Examorelin
Examorelin (INN) (developmental code names EP-23905, MF-6003), also known as hexarelin, is a potent, synthetic, peptidic, orally-active, centrally-penetrant, and highly selective agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) and a growth hormone secretagogue which was developed by . It is a hexapeptide with the amino acid sequence His-D-2-methyl-Trp-Ala-Trp-D-Phe-Lys-NH2 which was derived from GHRP-6. These GH-releasing peptides have no sequence similarity to ghrelin, but mimic ghrelin by acting as agonists at the ghrelin receptor.
primaryTopic
Examorelin
Examorelin (INN) (developmental code names EP-23905, MF-6003), also known as hexarelin, is a potent, synthetic, peptidic, orally-active, centrally-penetrant, and highly selective agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) and a growth hormone secretagogue which was developed by . It is a hexapeptide with the amino acid sequence His-D-2-methyl-Trp-Ala-Trp-D-Phe-Lys-NH2 which was derived from GHRP-6. These GH-releasing peptides have no sequence similarity to ghrelin, but mimic ghrelin by acting as agonists at the ghrelin receptor.
has abstract
Examorelin (INN) (developmenta ...... opment and was never marketed.
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CAS number
140703-51-1
ChEMBL
FDA UNII code
09QF37C617
PubChem
Wikipage page ID
46,963,951
page length (characters) of wiki page
Wikipage revision ID
993,029,186
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ATC prefix
None
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CAS number
ChEMBL
ChemSpiderID
elimination half-life
IUPAC name
IUPHAR ligand
PubChem
routes of administration
SMILES
CC1=CC[C@H]NC[C@H]N
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StdInChIKey
RVWNMGKSNGWLOL-GIIHNPQRSA-N
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synonyms
(L)-Histidyl-2-methyl-(D)-tryp ...... D)-phenylalanyl-(L)-lysinamide
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wikiPageUsesTemplate
subject
comment
Examorelin (INN) (developmenta ...... nists at the ghrelin receptor.
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label
Examorelin
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