From sensors to silencers: quinoline- and benzimidazole-sulfonamides as inhibitors for zinc proteases
about
Potent inhibition of dinuclear zinc(II) peptidase, an aminopeptidase from Aeromonas proteolytica, by 8-quinolinol derivatives: inhibitor design based on Zn2+ fluorophores, kinetic, and X-ray crystallographic studyMetalloprotein–Inhibitor Binding: Human Carbonic Anhydrase II as a Model for Probing Metal–Ligand Interactions in a Metalloprotein Active SiteA Noncompetitive Inhibitor for Mycobacterium tuberculosis ’s Class IIa Fructose 1,6-Bisphosphate AldolaseIdentifying chelators for metalloprotein inhibitors using a fragment-based approach.Investigation of self-immolative linkers in the design of hydrogen peroxide activated metalloprotein inhibitors.Exploring the influence of the protein environment on metal-binding pharmacophores.Emerging trends in metalloprotein inhibition.Morphological tuning via structural modulations in AIE luminogens with the minimum number of possible variables and their use in live cell imaging.From Zn to Mn: the study of novel manganese-binding groups in the search for new drugs against tuberculosis.Illuminating metal-ion sensors: benzimidazolesulfonamide metal complexes.A Bioinorganic Approach to Fragment-Based Drug Discovery Targeting Metalloenzymes.Dipicolinic Acid Derivatives as Inhibitors of New Delhi Metallo-β-lactamase-1.Synthesis of thieno[2,3-b]quinoline and selenopheno[2,3-b]quinoline derivatives via iodocyclization reaction and a DFT mechanistic study.Synthesis of Functionalized Quinolines through a Reaction of Amides and Alkynes Promoted by Triflic Anhydride/Pyridine.N-Heterocyclic carbene (NHC)-modulated Pd/Cu cocatalyzed three-component synthesis of 2,6-diarylquinolines.5-Position-selective C-H trifluoromethylation of 8-aminoquinoline derivatives.A general method for the metal-free, regioselective, remote C-H halogenation of 8-substituted quinolines.Targeting DNA Binding for NF-κB as an Anticancer Approach in Hepatocellular CarcinomaPalladium-catalyzed synthesis of polysubstituted quinolines from 2-amino aromatic ketones and alkynes
P2860
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P2860
From sensors to silencers: quinoline- and benzimidazole-sulfonamides as inhibitors for zinc proteases
description
2010 nî lūn-bûn
@nan
2010 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
From sensors to silencers: qui ...... inhibitors for zinc proteases
@ast
From sensors to silencers: qui ...... inhibitors for zinc proteases
@en
From sensors to silencers: qui ...... inhibitors for zinc proteases.
@nl
type
label
From sensors to silencers: qui ...... inhibitors for zinc proteases
@ast
From sensors to silencers: qui ...... inhibitors for zinc proteases
@en
From sensors to silencers: qui ...... inhibitors for zinc proteases.
@nl
prefLabel
From sensors to silencers: qui ...... inhibitors for zinc proteases
@ast
From sensors to silencers: qui ...... inhibitors for zinc proteases
@en
From sensors to silencers: qui ...... inhibitors for zinc proteases.
@nl
P2093
P2860
P356
P1476
From sensors to silencers: qui ...... inhibitors for zinc proteases
@en
P2093
Arpita Agrawal
César Augusto F de Oliveira
Matthieu Rouffet
P2860
P304
P356
10.1021/JA101088J
P407
P577
2010-06-01T00:00:00Z