Nuclear hormone receptors: ligand-activated regulators of transcription and diverse cell responses.
about
Estrogen receptor transcription and transactivation: Basic aspects of estrogen action.A peroxisome proliferator-activated receptor gamma ligand inhibits adipocyte differentiationCrystal structure of a mutant hERalpha ligand-binding domain reveals key structural features for the mechanism of partial agonismCrystallographic comparison of the estrogen and progesterone receptor's ligand binding domainsInCHlib – interactive cluster heatmap for web applicationsGeneration and reproductive phenotypes of mice lacking estrogen receptor betaMolecular determinants of tissue selectivity in estrogen receptor modulators.Discovering small-molecule estrogen receptor α/coactivator binding inhibitors: high-throughput screening, ligand development, and models for enhanced potency.Ligand-protein interactions in nuclear receptors of hormones.Protein and RNA engineering to customize microbial molecular reporting.N-arylbenzamides: extremely simple scaffolds for the development of novel estrogen receptor agonists.Bibenzyl- and stilbene-core compounds with non-polar linker atom substituents as selective ligands for estrogen receptor beta.Phenethyl pyridines with non-polar internal substituents as selective ligands for estrogen receptor beta.JNK suppression is essential for 17β-Estradiol inhibits prostaglandin E2-Induced uPA and MMP-9 expressions and cell migration in human LoVo colon cancer cells.Glucocorticoids repress NF-kappaB-driven genes by disturbing the interaction of p65 with the basal transcription machinery, irrespective of coactivator levels in the cellFluorine-substituted cyclofenil derivatives as estrogen receptor ligands: synthesis and structure-affinity relationship study of potential positron emission tomography agents for imaging estrogen receptors in breast cancer.Ethnic variation in allele distribution of the androgen receptor (AR) (CAG)n repeat.Toxicological mechanism of endocrine disrupting chemicals:is estrogen receptor involved?AR inhibitors identified by high-throughput microscopy detection of conformational change and subcellular localization.Improving selective androgen receptor modulator discovery and preclinical evaluation.Analysis of estrogen receptor interaction with a repressor of estrogen receptor activity (REA) and the regulation of estrogen receptor transcriptional activity by REA.Why (multi)targeting of cyclin-dependent kinases is a promising therapeutic option for hormone-positive breast cancer and beyond.The olive oil phenolic (-)-oleocanthal modulates estrogen receptor expression in luminal breast cancer in vitro and in vivo and synergizes with tamoxifen treatment.Study on cytochrome p-450 dependent retinoic Acid metabolism and its inhibitors as potential agents for cancer therapy.Interference with ER-α enhances the therapeutic efficacy of the selective CDK inhibitor roscovitine towards ER-positive breast cancer cells.Rodent Models of Non-classical Progesterone Action Regulating Ovulation.Roscovitine, a selective CDK inhibitor, reduces the basal and estrogen-induced phosphorylation of ER-α in human ER-positive breast cancer cells.Fatty acid binding profile of the liver X receptor α.Fluorescent cellular sensors of steroid receptor ligands.Directed evolution of human estrogen receptor variants with significantly enhanced androgen specificity and affinity.Phosphorylation of thyroid hormone receptors by protein kinase A regulates DNA recognition by specific inhibition of receptor monomer binding.Fertility and developmental toxicity assessment in rats and rabbits with LY500307, a selective estrogen receptor beta (ERβ) agonist.Regulation of bcl-2 transcription by estrogen receptor-α and c-Jun in human endometrium.p38α MAPK mediates 17β-estradiol inhibition of MMP-2 and -9 expression and cell migration in human lovo colon cancer cells.Controversial effect on Erk activation of some cytotoxic drugs in human LOVO colon cancer cells.
P2860
Q24800814-CB863764-DF31-40F2-98DA-7312D7FCF660Q27618352-401EDD98-027C-4FD8-90FA-529BA8CDE53BQ27630889-838772A7-7AF5-4132-A248-3CBB88F24209Q27757822-06B0B14F-E872-4897-8E0F-D9E8DFA54771Q27902279-27EAFB21-D517-4905-9B99-19563E812DECQ28513765-C60D2505-4A67-43F0-AD38-920CED01A61AQ33747238-4D5B8BFF-D029-41D0-AAF0-538AEE4B0A61Q33834493-13399ECC-28F2-4843-BC5C-EB6D9CAE6E72Q33957129-8852DB58-4C6C-42DD-A18E-E96317B47297Q34059491-9095ABC7-A403-4DA7-9466-3A09A1ABD602Q34101025-0F5D05D7-A987-4EC2-84BE-5B3A5A56D282Q35220167-D7E59101-AF59-4EEA-BF2D-EB2EB4C0324AQ35222159-D091885D-D5E9-4636-BDAE-9B8B82E9A6ABQ35232048-C792F919-0DAB-4F60-99D6-B0714B4646C6Q35666145-66E5D2A3-9119-4360-9AA2-6A2031D65FBDQ36848788-28749149-76DC-4E6B-A5C6-CE8ADBE92ECEQ37323212-7E17C67B-AB33-491E-8530-CCED1486A75AQ37326623-D7D29371-A95E-4889-9E38-DB10838E508DQ37418519-22ADA038-6348-465B-93AE-96C9A56A7FE1Q38088367-843A26C4-2EB5-485A-9BFB-A0C4F8B00C44Q38308965-7E509606-EFCA-463C-99D2-14297ABD4715Q38675849-B2E9E277-1C04-4DC7-9D91-62BB9C645187Q38699970-10222A34-4C69-4E19-85B2-C974AD1F32EBQ39281494-A2A91E98-8B0F-4B4B-9BE5-67608563DB51Q39594930-1AFCD041-20AC-411A-B246-5F9BA4107D56Q41097262-7D77BF1B-5F1C-418B-936E-D7DCAE86F3DDQ42484098-C6B707F3-5A8E-40EA-91B1-B3E4C0FFBEA3Q43089720-79592751-1B9A-416C-8E23-31605BDD6EE7Q44578576-7E190830-B160-43CE-8C92-98690E55574AQ44907820-4801603A-8846-4184-957A-C71146E2A45BQ46081560-C8449137-028F-4C63-B4EF-C2F53077B9B4Q46318067-3ED7B729-5210-4273-8F57-F880C9F9220EQ46361342-E8E49347-EE18-430D-B1B4-63F200383431Q53182315-D380D193-6E39-49C6-B70C-2F66497E061CQ55070462-9B1C9D34-16AA-4BE0-8EC6-8802F62C9617
P2860
Nuclear hormone receptors: ligand-activated regulators of transcription and diverse cell responses.
description
1996 nî lūn-bûn
@nan
1996年の論文
@ja
1996年論文
@yue
1996年論文
@zh-hant
1996年論文
@zh-hk
1996年論文
@zh-mo
1996年論文
@zh-tw
1996年论文
@wuu
1996年论文
@zh
1996年论文
@zh-cn
name
Nuclear hormone receptors: lig ...... on and diverse cell responses.
@en
type
label
Nuclear hormone receptors: lig ...... on and diverse cell responses.
@en
prefLabel
Nuclear hormone receptors: lig ...... on and diverse cell responses.
@en
P1476
Nuclear hormone receptors: lig ...... on and diverse cell responses.
@en
P2093
Katzenellenbogen BS
Katzenellenbogen JA
P304
P356
10.1016/S1074-5521(96)90143-X
P577
1996-07-01T00:00:00Z