A heterodimer-selective agonist shows in vivo relevance of G protein-coupled receptor dimers.
about
Cys-27 variant of human δ-opioid receptor modulates maturation and cell surface delivery of Phe-27 variant via heteromerizationThe G protein-coupled receptor heterodimer network (GPCR-HetNet) and its hub componentsClinically employed opioid analgesics produce antinociception via μ-δ opioid receptor heteromers in Rhesus monkeysHeteromerization of G protein-coupled receptors: relevance to neurological disorders and neurotherapeutics.The δ opioid receptor agonist SNC80 selectively activates heteromeric μ-δ opioid receptorsStandard opioid agonists activate heteromeric opioid receptors: evidence for morphine and [d-Ala(2)-MePhe(4)-Glyol(5)]enkephalin as selective μ-δ agonistsReceptor heteromerization and drug discovery.Allostery at G protein-coupled receptor homo- and heteromers: uncharted pharmacological landscapesUnidirectional cross-activation of GRPR by MOR1D uncouples itch and analgesia induced by opioidsBuilding a new conceptual framework for receptor heteromersG-protein-coupled receptor heteromers: function and ligand pharmacologyBasic Pharmacological and Structural Evidence for Class A G-Protein-Coupled Receptor HeteromerizationAntibodies to probe endogenous G protein-coupled receptor heteromer expression, regulation, and functionNeuroprotective mechanisms of the ACE2-angiotensin-(1-7)-Mas axis in strokeOpioid receptors: toward separation of analgesic from undesirable effectsKir3 channel signaling complexes: focus on opioid receptor signalingBiological redundancy of endogenous GPCR ligands in the gut and the potential for endogenous functional selectivityMolecular switches of the κ opioid receptor triggered by 6'-GNTI and 5'-GNTI.Preferred supramolecular organization and dimer interfaces of opioid receptors from simulated self-associationCircadian-related heteromerization of adrenergic and dopamine D₄ receptors modulates melatonin synthesis and release in the pineal glandAnti-analgesic effect of the mu/delta opioid receptor heteromer revealed by ligand-biased antagonismCrosstalk between GABAB and mGlu1a receptors reveals new insight into GPCR signal integrationA bivalent ligand (KMN-21) antagonist for mu/kappa heterodimeric opioid receptorsStructure-guided development of heterodimer-selective GPCR ligandsActivation of G protein-coupled receptors: beyond two-state models and tertiary conformational changes.Transmembrane domain IV of the Gallus gallus VT2 vasotocin receptor is essential for forming a heterodimer with the corticotrophin releasing hormone receptorRegulation of neuronal pH by the metabotropic Zn(2+)-sensing Gq-coupled receptor, mZnR/GPR39.Apelin receptor homodimer-oligomers revealed by single-molecule imaging and novel G protein-dependent signaling.Identification of the First Marine-Derived Opioid Receptor "Balanced" Agonist with a Signaling Profile That Resembles the EndorphinsRequirements and ontology for a G protein-coupled receptor oligomerization knowledge base.Direct interaction of GABAB receptors with M2 muscarinic receptors enhances muscarinic signaling.Endothelin receptors: what's new and what do we need to know?An in vivo demonstration of functional G protein-coupled receptor dimers.Increasingly accurate dynamic molecular models of G-protein coupled receptor oligomers: Panacea or Pandora's box for novel drug discovery?Search for the "ideal analgesic" in pain treatment by engineering the mu-opioid receptor.Dynamic models of G-protein coupled receptor dimers: indications of asymmetry in the rhodopsin dimer from molecular dynamics simulations in a POPC bilayer.Contribution of mu and delta opioid receptors to the pharmacological profile of kappa opioid receptor subtypes.Diversifying the repertoire of G protein-coupled receptors through oligomerization.Seven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery.Opioid-receptor-heteromer-specific trafficking and pharmacology.
P2860
Q24300182-5A0E486E-3652-460A-8376-EC4E9CA37AEDQ24564171-4B8AB665-786E-436B-A315-99CCB8C5FA2EQ24597777-DC62D448-6A49-497E-8CF4-CBD08724CC8DQ24630645-4194CB93-88D7-437F-A849-91CF0074018CQ24630886-DA2E85E3-20EB-41BC-8FBF-0FCE2952EEC3Q24631212-3C8C8215-5D8E-420E-A8DC-B2D807532019Q24631740-84581E51-B677-4E14-B58B-FE13AD2D9871Q24633877-4049209A-0BDF-4AD7-A846-8F99E7679B5CQ24634901-28882711-E31A-47A3-9F0E-71756249B078Q24644975-DF5CF8B6-5270-48EA-9BD3-3C60827C9977Q24653717-E4BC2D51-970E-4AD5-A236-97F806760569Q26749791-7DCEDC8C-5895-4F1F-8FE7-20C359D84875Q26992192-4269409C-E27C-4D7C-BA93-52E6A50E3DBEQ26998948-227B2272-155B-44CD-B45A-AE8012B69ECAQ27002925-820BB6A0-AA09-4E2A-B702-009E08DA4569Q27006957-5593246E-40F3-4E71-9F5C-91B9191717E7Q27021347-766D6420-185A-4DE4-AAA2-FCC8CC4C74F4Q27302413-9D9AC060-1C90-4628-A102-1A5A6C46C069Q27319797-502825A5-EDCA-45E1-BC71-83CCAE992A12Q28480542-97B12DEA-33EE-448C-941D-9C85FA1483BDQ28488120-079C191E-C1BA-44C5-9DA7-8EB34E1B4BAEQ28564967-971A6E51-CE63-4FD6-9BF0-457E17B13ED6Q28822182-86F3792E-98B5-46EF-9141-CEAC9474CD60Q28828634-48B61062-6FCE-4FC3-AA45-2406CB2ADC20Q30364526-04BDB85F-3E3B-4B47-8FED-4871A5FC556DQ30413870-2E71F9F0-30F7-4AFB-93C0-A3601E0B1C3DQ30665208-96206559-CB2C-430A-AFBE-BD3BD26A048CQ30835080-6D299982-51F7-4B89-BDB5-9F7C7C506E42Q30841944-DB0B386F-FAF4-469E-BA3E-AB48C7D36715Q33286209-5225AE0E-FD03-493C-BD2E-25EEAD2D8FFEQ33637415-844F6F60-BB98-491A-9695-A289D3B6D660Q33686555-994C42B4-9935-44A6-8EE2-29DBC7933DA3Q33720008-BF15964F-7648-4AB7-936F-4E60DB43DF35Q33767121-248F7EA2-1C64-4BE9-BDCC-10C5B83B9C27Q33807778-E66B275C-767E-42CD-A707-BB253A888272Q33825866-9CBCC762-A9E9-47E9-B1C5-0627571BDE1DQ33863139-2ABC34B4-6857-47C4-A470-9904C87C607CQ33863332-D8DEC747-B0FA-412F-96AC-E38B90CCC6B4Q33890786-E58D9DF4-A66D-40EA-9EA1-8201A9098642Q33978499-8C629CE8-40DE-45DC-962F-7F9A4A96FAE0
P2860
A heterodimer-selective agonist shows in vivo relevance of G protein-coupled receptor dimers.
description
2005 nî lūn-bûn
@nan
2005 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2005年の論文
@ja
2005年論文
@yue
2005年論文
@zh-hant
2005年論文
@zh-hk
2005年論文
@zh-mo
2005年論文
@zh-tw
2005年论文
@wuu
name
A heterodimer-selective agonis ...... rotein-coupled receptor dimers
@nl
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@ast
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en-gb
type
label
A heterodimer-selective agonis ...... rotein-coupled receptor dimers
@nl
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@ast
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en-gb
prefLabel
A heterodimer-selective agonis ...... rotein-coupled receptor dimers
@nl
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@ast
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en-gb
P2093
P2860
P3181
P356
P1476
A heterodimer-selective agonis ...... otein-coupled receptor dimers.
@en
P2093
Evi Kostenis
Jamie Fong
Jennifer L Whistler
Maria Waldhoer
Mary M Lunzer
Philip S Portoghese
Robert M Jones
Shiv K Sharma
P2860
P304
P3181
P356
10.1073/PNAS.0501112102
P407
P577
2005-06-02T00:00:00Z