G-protein-coupled receptor heterodimerization modulates receptor function
about
GPCR oligomers in pharmacology and signalingMetabotropic glutamate mGlu2 receptor is necessary for the pharmacological and behavioral effects induced by hallucinogenic 5-HT2A receptor agonistsCys-140 is critical for metabotropic glutamate receptor-1 dimerizationHeterodimerization of alpha 2A- and beta 1-adrenergic receptorsCys-27 variant of human δ-opioid receptor modulates maturation and cell surface delivery of Phe-27 variant via heteromerizationIdentification and pharmacological characterization of the prostaglandin FP receptor and FP receptor variant complexesA heterodimer-selective agonist shows in vivo relevance of G protein-coupled receptor dimers.Evidence for a single heptahelical domain being turned on upon activation of a dimeric GPCRClinically employed opioid analgesics produce antinociception via μ-δ opioid receptor heteromers in Rhesus monkeysHeterodimerization of V1a and V2 vasopressin receptors determines the interaction with beta-arrestin and their trafficking patternsHeteromeric association creates a P2Y-like adenosine receptorFunctional crosstalk and heteromerization of serotonin 5-HT2A and dopamine D2 receptorsHeteromerization of G protein-coupled receptors: relevance to neurological disorders and neurotherapeutics.The δ opioid receptor agonist SNC80 selectively activates heteromeric μ-δ opioid receptorsStandard opioid agonists activate heteromeric opioid receptors: evidence for morphine and [d-Ala(2)-MePhe(4)-Glyol(5)]enkephalin as selective μ-δ agonistsReceptor heteromerization and drug discovery.Allostery at G protein-coupled receptor homo- and heteromers: uncharted pharmacological landscapesUnidirectional cross-activation of GRPR by MOR1D uncouples itch and analgesia induced by opioidsMarked changes in signal transduction upon heteromerization of dopamine D1 and histamine H3 receptorsPharmacological characterization of the human 5-HT(4(d)) receptor splice variant stably expressed in Chinese hamster ovary cellsNeuropathic Pain due to Small Fiber Neuropathy in Aging: Current Management and Future ProspectsDynorphin--still an extraordinarily potent opioid peptideNovel GPCR paradigms at the μ-opioid receptorLipid- and sugar-modified endomorphins: novel targets for the treatment of neuropathic painAntibodies to probe endogenous G protein-coupled receptor heteromer expression, regulation, and functionOpioid receptors: toward separation of analgesic from undesirable effectsOpioid receptor heteromers in analgesiaKir3 channel signaling complexes: focus on opioid receptor signalingDopamine-induced plasticity, phospholipase D (PLD) activity and cocaine-cue behavior depend on PLD-linked metabotropic glutamate receptors in amygdalaCrystal structure of the µ-opioid receptor bound to a morphinan antagonistMembrane-Mediated Oligomerization of G Protein Coupled Receptors and Its Implications for GPCR FunctionExport from the endoplasmic reticulum represents the limiting step in the maturation and cell surface expression of the human delta opioid receptorFunctional characterization of mutations in melanocortin-4 receptor associated with human obesityHeterodimerization of mu and delta opioid receptors: A role in opiate synergySelective interactions between helix VIII of the human mu-opioid receptors and the C terminus of periplakin disrupt G protein activationHypersensitization of the Orexin 1 receptor by the CB1 receptor: evidence for cross-talk blocked by the specific CB1 antagonist, SR141716Oligomerization of G-protein-coupled receptors shown by selective co-immunoprecipitationDimerization and phosphorylation of thyrotropin-releasing hormone receptors are modulated by agonist stimulationMu and Delta opioid receptors activate the same G proteins in human neuroblastoma SH-SY5Y cellsOligomerization of opioid receptors with beta 2-adrenergic receptors: a role in trafficking and mitogen-activated protein kinase activation
P2860
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P2860
G-protein-coupled receptor heterodimerization modulates receptor function
description
1999 nî lūn-bûn
@nan
1999 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի հունիսին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
G-protein-coupled receptor heterodimerization modulates receptor function
@ast
G-protein-coupled receptor heterodimerization modulates receptor function
@en
G-protein-coupled receptor heterodimerization modulates receptor function
@nl
type
label
G-protein-coupled receptor heterodimerization modulates receptor function
@ast
G-protein-coupled receptor heterodimerization modulates receptor function
@en
G-protein-coupled receptor heterodimerization modulates receptor function
@nl
prefLabel
G-protein-coupled receptor heterodimerization modulates receptor function
@ast
G-protein-coupled receptor heterodimerization modulates receptor function
@en
G-protein-coupled receptor heterodimerization modulates receptor function
@nl
P2860
P3181
P356
P1433
P1476
G-protein-coupled receptor heterodimerization modulates receptor function
@en
P2093
P2860
P2888
P304
P3181
P356
10.1038/21441
P407
P577
1999-06-17T00:00:00Z
P5875
P6179
1000614717