Development of Selective Inhibitors for Aldehyde Dehydrogenases Based on Substituted Indole-2,3-diones
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Structural, Biochemical, and Computational Studies Reveal the Mechanism of Selective Aldehyde Dehydrogenase 1A1 Inhibition by Cytotoxic Duocarmycin AnaloguesPharmacological recruitment of aldehyde dehydrogenase 3A1 (ALDH3A1) to assist ALDH2 in acetaldehyde and ethanol metabolism in vivo.Discovery of a series of aromatic lactones as ALDH1/2-directed inhibitors.Substrate Specificity, Inhibitor Selectivity and Structure-Function Relationships of Aldo-Keto Reductase 1B15: A Novel Human Retinaldehyde Reductase.Discovery of Novel Isatin-Based p53 InducersA High-Content Assay Enables the Automated Screening and Identification of Small Molecules with Specific ALDH1A1-Inhibitory Activity.Discovery of NCT-501, a Potent and Selective Theophylline-Based Inhibitor of Aldehyde Dehydrogenase 1A1 (ALDH1A1)Aldehyde dehydrogenases in cancer stem cells: potential as therapeutic targets.Targeting aldehyde dehydrogenase activity in head and neck squamous cell carcinoma with a novel small molecule inhibitorAldehyde dehydrogenase 1A1 increases NADH levels and promotes tumor growth via glutathione/dihydrolipoic acid-dependent NAD+ reduction.Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors.Discovery of Orally Bioavailable, Quinoline-based Aldehyde Dehydrogenase 1A1 (ALDH1A1) Inhibitors with Potent Cellular Activity.
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P2860
Development of Selective Inhibitors for Aldehyde Dehydrogenases Based on Substituted Indole-2,3-diones
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2014 nî lūn-bûn
@nan
2014 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@ast
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@en
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@nl
type
label
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@ast
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@en
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@nl
prefLabel
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@ast
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@en
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@nl
P2093
P2860
P356
P1476
Development of Selective Inhib ...... Substituted Indole-2,3-diones
@en
P2093
Bibek Parajuli
Che-Hong Chen
Daria Mochly-Rosen
P2860
P304
P356
10.1021/JM401377V
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P577
2014-02-13T00:00:00Z