The novel isoxazoline ectoparasiticide fluralaner: selective inhibition of arthropod γ-aminobutyric acid- and L-glutamate-gated chloride channels and insecticidal/acaricidal activity.
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Efficacy of orally administered fluralaner (Bravecto™) or topically applied imidacloprid/moxidectin (Advocate®) against generalized demodicosis in dogsSystemically and cutaneously distributed ectoparasiticides: a review of the efficacy against ticks and fleas on dogsComparative efficacy of oral administrated afoxolaner (NexGard™) and fluralaner (Bravecto™) with topically applied permethrin/imidacloprid (Advantix(®)) against transmission of Ehrlichia canis by infected Rhipicephalus sanguineus ticks to dogs.Fluralaner, a novel isoxazoline, prevents flea (Ctenocephalides felis) reproduction in vitro and in a simulated home environment.Molecular cloning and characterization of a glycine-like receptor gene from the cattle tick Rhipicephalus (Boophilus) microplus (Acari: Ixodidae).The speed of kill of fluralaner (Bravecto™) against Ixodes ricinus ticks on dogs.Onset of activity of fluralaner (BRAVECTO™) against Ctenocephalides felis on dogs.Fluralaner activity against life stages of ticks using Rhipicephalus sanguineus and Ornithodoros moubata IN in vitro contact and feeding assaysA quantitative evaluation of the extent of fluralaner uptake by ticks (Ixodes ricinus, Ixodes scapularis) in fluralaner (Bravecto) treated vs. untreated dogs using the parameters tick weight and coxal index.A novel combination of fipronil and permethrin (Frontline Tri-Act®/Frontect®) reduces risk of transmission of Babesia canis by Dermacentor reticulatus and of Ehrlichia canis by Rhipicephalus sanguineus ticks to dogs.Comparative pharmacokinetics of fluralaner in dogs and cats following single topical or intravenous administrationEfficacy of fluralaner spot-on solution against induced infestations with Rhipicephalus sanguineus on dogsEvaluation of fluralaner and afoxolaner treatments to control flea populations, reduce pruritus and minimize dermatologic lesions in naturally infested dogs in private residences in west central Florida USAMosquitocidal Activity and Mode of Action of the Isoxazoline FluralanerPharmacokinetics of fluralaner in dogs following a single oral or intravenous administration.A randomized, blinded, controlled and multi-centered field study comparing the efficacy and safety of Bravecto (fluralaner) against Frontline (fipronil) in flea- and tick-infested dogs.Isoxazolines: A Novel Chemotype Highly Effective on Ectoparasites.Systemic insecticide treatment of the canine reservoir of Trypanosoma cruzi induces high levels of lethality in Triatoma infestans, a principal vector of Chagas disease.From the Cover: Functional Analysis Reveals Glutamate and Gamma-Aminobutyric Acid-Gated Chloride Channels as Targets of Avermectins in the Carmine Spider Mite.Comparative in vitro evaluation of contact activity of fluralaner, spinosad, phoxim, propoxur, permethrin and deltamethrin against the northern fowl mite, Ornithonyssus sylviarum.Safety of fluralaner oral solution, a novel systemic antiparasitic treatment for chickens, in laying hens after oral administration via drinking water.Field efficacy and safety of fluralaner solution for administration in drinking water for the treatment of poultry red mite (Dermanyssus gallinae) infestations in commercial flocks in EuropeThe intravenous and oral pharmacokinetics of lotilaner in dogs.The novel isoxazoline ectoparasiticide lotilaner (Credelio™): a non-competitive antagonist specific to invertebrates γ-aminobutyric acid-gated chloride channels (GABACls).A G326E substitution in the glutamate-gated chloride channel 3 (GluCl3) of the two-spotted spider mite Tetranychus urticae abolishes the agonistic activity of macrocyclic lactones.Safety evaluation of lotilaner in dogs after oral administration as flavoured chewable tablets (Credelio™).The Biology and Ecology of Cat Fleas and Advancements in Their Pest Management: A Review.The acaricidal speed of kill of orally administered fluralaner against poultry red mites (Dermanyssus gallinae) on laying hens and its impact on mite reproduction.Safety of fluralaner oral solution, a novel systemic poultry red mite treatment, for chicken breeders' reproductive performances.Afoxolaner and fluralaner treatment do not impact on cutaneous Demodex populations of healthy dogs.Efficacy and safety assessment of a water-soluble formulation of fluralaner for treatment of natural Ornithonyssus sylviarum infestations in laying hens.Catalytic enantioselective synthesis of carboxy-substituted 2-isoxazolines by cascade oxa-Michael-cyclization.Efficacy of fluralaner in 17 dogs with sarcoptic mange.The use of oral fluralaner for the treatment of feline generalised demodicosis: a case report.Access to benzo-fused nine-membered heterocyclic alkenes with a trifluoromethyl carbinol moiety via a double decarboxylative formal ring-expansion process under palladium catalysis.In vitro activity of fluralaner and commonly used acaricides against Dermanyssus gallinae isolates from Europe and Brazil.Safety of lotilaner flavoured chewable tablets (CredelioTM) after oral administration in cats.The fungal alkaloid Okaramine-B activates an L-glutamate-gated chloride channel from Ixodes scapularis, a tick vector of Lyme disease.Pharmacokinetics of lotilaner following a single oral or intravenous administration in cats.Repurposing isoxazoline veterinary drugs for control of vector-borne human diseases
P2860
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P2860
The novel isoxazoline ectoparasiticide fluralaner: selective inhibition of arthropod γ-aminobutyric acid- and L-glutamate-gated chloride channels and insecticidal/acaricidal activity.
description
2013 nî lūn-bûn
@nan
2013 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@ast
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@en
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@nl
type
label
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@ast
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@en
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@nl
prefLabel
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@ast
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@en
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@nl
P2093
P1476
The novel isoxazoline ectopara ...... ecticidal/acaricidal activity.
@en
P2093
Christian Wolf
Heike Williams
Michael Gassel
Sandra Noack
Thomas Ilg
P304
P356
10.1016/J.IBMB.2013.11.009
P577
2013-12-21T00:00:00Z