Novel non-active site inhibitor of Cryptosporidium hominis TS-DHFR identified by a virtual screen
about
First Three-Dimensional Structure of Toxoplasma gondii Thymidylate Synthase–Dihydrofolate Reductase: Insights for Catalysis, Interdomain Interactions, and Substrate ChannelingExploring novel strategies for AIDS protozoal pathogens: α-helix mimetics targeting a key allosteric protein–protein interaction in C. hominis thymidylate synthase-dihydrofolate reductase (TS-DHFR)Integrated text mining and chemoinformatics analysis associates diet to health benefit at molecular levelProdrug activation by Cryptosporidium thymidine kinase.Virtual screening reveals allosteric inhibitors of the Toxoplasma gondii thymidylate synthase-dihydrofolate reductaseUnderstanding the molecular mechanism of substrate channeling and domain communication in protozoal bifunctional TS-DHFR.Selective peptide inhibitors of bifunctional thymidylate synthase-dihydrofolate reductase from Toxoplasma gondii provide insights into domain-domain communication and allosteric regulation.Synthesis and biological evaluation of biguanide and dihydrotriazine derivatives as potential inhibitors of dihydrofolate reductase of opportunistic microorganisms.
P2860
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P2860
Novel non-active site inhibitor of Cryptosporidium hominis TS-DHFR identified by a virtual screen
description
2008 nî lūn-bûn
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2008年の論文
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2008年学术文章
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2008年学术文章
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2008年学术文章
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2008年学术文章
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2008年学术文章
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2008年學術文章
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2008年學術文章
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2008年學術文章
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name
Novel non-active site inhibito ...... identified by a virtual screen
@en
Novel non-active site inhibito ...... dentified by a virtual screen.
@nl
type
label
Novel non-active site inhibito ...... identified by a virtual screen
@en
Novel non-active site inhibito ...... dentified by a virtual screen.
@nl
prefLabel
Novel non-active site inhibito ...... identified by a virtual screen
@en
Novel non-active site inhibito ...... dentified by a virtual screen.
@nl
P2093
P2860
P1476
Novel non-active site inhibito ...... identified by a virtual screen
@en
P2093
Chloe Atreya
Karen S Anderson
Marina Udier-Blagovic
Melissa A Vargo
Oladapo Babatunde
W Edward Martucci
P2860
P304
P356
10.1016/J.BMCL.2008.11.054
P407
P577
2008-11-20T00:00:00Z