2-Naphthalenesulphonyl L-aspartyl-(2-phenethyl)amide (2-NAP)--a selective cholecystokinin CCKA-receptor antagonist
about
Characterization of the binding of a novel radioligand to CCKB/gastrin receptors in membranes from rat cerebral cortexEffects of peripheral CCK receptor blockade on feeding responses to duodenal nutrient infusions in ratsCholecystokinin antagonists: pharmacological and therapeutic potential.Molecular cloning, expression and pharmacological characterization of the canine cholecystokinin 1 receptorPEGylated cholecystokinin prolongs satiation in rats: dose dependency and receptor involvement.Unexpected relationship between plasma protein binding and the pharmacodynamics of 2-NAP, a CCK1-receptor antagonist.PEGylated cholecystokinin is more potent in inducing anorexia than conditioned taste aversion in rats.Analysis of variation in L-365,260 competition curves in radioligand binding assays2-Naphthalenesulphanyl-L-aspartyl-2-(phenethyl) amide (2-NAP) and food intake in rats: evidence that endogenous peripheral CCK does not play a major role as a satiety factor.Pharmacological evidence for putative CCK(1) receptor heterogeneity in human colon smooth muscle.Effects of peripheral CCK receptor blockade on food intake in rats.Relative blood-brain barrier permeabilities of the cholecystokinin receptor antagonists devazepide and A-65186 in rats.Cholecystokinin-A receptor antagonists: therapies for gastrointestinal disorders.
P2860
Q28343282-24E24B8A-48A8-421D-9432-661F64E6BCDAQ28578998-B1B80F26-4F11-4858-8F98-044EF13E9475Q34203535-DDB0582D-6515-4E51-9ABC-11E709947E1CQ35048902-BB05EC68-50A5-4077-87BA-09EC18F017BBQ36094371-C129F0F4-2EE5-4C1C-8F35-FD31B28A0CE5Q38508311-1C7960E5-C9CB-4A72-A4CE-63BED6A01F61Q41810707-CE7F66AE-8DD7-4A58-9E3F-C195C648E78EQ41823935-C431C894-96A7-4452-9FF3-778371848B54Q41903306-5477198E-6DC0-423D-943F-55E644F7F769Q43263725-2968045A-1F2E-4F88-8707-22A91EFB9540Q44435084-B63CC35C-E03B-4D5B-8740-015A08209A43Q48102294-FA49C9C7-D81A-4EE6-A362-541421EE60AAQ48660973-5368BA6A-FD2C-44B4-A18B-02B18ACB405C
P2860
2-Naphthalenesulphonyl L-aspartyl-(2-phenethyl)amide (2-NAP)--a selective cholecystokinin CCKA-receptor antagonist
description
1993 nî lūn-bûn
@nan
1993年の論文
@ja
1993年論文
@yue
1993年論文
@zh-hant
1993年論文
@zh-hk
1993年論文
@zh-mo
1993年論文
@zh-tw
1993年论文
@wuu
1993年论文
@zh
1993年论文
@zh-cn
name
2-Naphthalenesulphonyl L-aspar ...... kinin CCKA-receptor antagonist
@en
type
label
2-Naphthalenesulphonyl L-aspar ...... kinin CCKA-receptor antagonist
@en
prefLabel
2-Naphthalenesulphonyl L-aspar ...... kinin CCKA-receptor antagonist
@en
P2093
P2860
P1476
2-Naphthalenesulphonyl L-aspar ...... kinin CCKA-receptor antagonist
@en
P2093
P2860
P304
P356
10.1111/J.1476-5381.1993.TB12870.X
P407
P577
1993-03-01T00:00:00Z