Structure-based design of a highly selective catalytic site-directed inhibitor of Ser/Thr protein phosphatase 2B (calcineurin).
about
Targeting protein serine/threonine phosphatases for drug developmentSites of protein kinase A activation of the human ClC-2 Cl(-) channelSynthesis and characterization of pseudocantharidins, novel phosphatase modulators that promote the inclusion of exon 7 into the SMN (survival of motoneuron) pre-mRNACrystallization and preliminary crystallographic study of a trypsin-resistant catalytic domain of human calcineurin.A cytoplasmic new catalytic subunit of calcineurin in Trypanosoma cruzi and its molecular and functional characterizationNovel inhibitors of the calcineurin/NFATc hub - alternatives to CsA and FK506?Norcantharidin, a protective therapeutic agent in renal tubulointerstitial fibrosis.Norcantharidin inhibits the expression of extracellular matrix and TGF-β1 in HK-2 cells induced by high glucose independent of calcineurin signal pathway.Effect of norcantharidin on proliferation and invasion of human gallbladder carcinoma GBC-SD cellsExploration of new drug-like inhibitors for serine/threonine protein phosphatase 5 of Plasmodium falciparum: a docking and simulation study.Indomethacin serves as a potential inhibitor of protein phosphatases.Facile Chemical Access to Biologically Active Norcantharidin Derivatives from Biomass.Chemoselective flow hydrogenation approaches to isoindole-7-carboxylic acids and 7-oxa-bicyclio[2.2.1]heptanes
P2860
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P2860
Structure-based design of a highly selective catalytic site-directed inhibitor of Ser/Thr protein phosphatase 2B (calcineurin).
description
2003 nî lūn-bûn
@nan
2003年の論文
@ja
2003年学术文章
@wuu
2003年学术文章
@zh
2003年学术文章
@zh-cn
2003年学术文章
@zh-hans
2003年学术文章
@zh-my
2003年学术文章
@zh-sg
2003年學術文章
@yue
2003年學術文章
@zh-hant
name
Structure-based design of a hi ...... phosphatase 2B (calcineurin).
@en
Structure-based design of a hi ...... Ser/Thr protein phosphatase 2B
@nl
type
label
Structure-based design of a hi ...... phosphatase 2B (calcineurin).
@en
Structure-based design of a hi ...... Ser/Thr protein phosphatase 2B
@nl
prefLabel
Structure-based design of a hi ...... phosphatase 2B (calcineurin).
@en
Structure-based design of a hi ...... Ser/Thr protein phosphatase 2B
@nl
P2093
P356
P1476
Structure-based design of a hi ...... phosphatase 2B (calcineurin).
@en
P2093
Mikiko Sodeoka
Naoto Tanohira
Nozomu Hirukawa
Yoshiyasu Baba
P304
P356
10.1021/JA034694Y
P407
P577
2003-08-01T00:00:00Z