Molecular basis for P-site inhibition of adenylyl cyclase
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Effect of Iboga alkaloids on µ-opioid receptor-coupled G protein activationCrystal structures of the catalytic domain of human soluble guanylate cyclasePAM mediates sustained inhibition of cAMP signaling by sphingosine-1-phosphateMolecular details of cAMP generation in mammalian cells: a tale of two systemsBacillus anthracis edema factor substrate specificity: evidence for new modes of actionSimilarly potent inhibition of adenylyl cyclase by P-site inhibitors in hearts from wild type and AC5 knockout miceStructural Basis for Inhibition of Mammalian Adenylyl Cyclase by Calcium †Structural and functional analysis of the Lmo2642 cyclic nucleotide phosphodiesterase from Listeria monocytogenesStructure of the Cmr2 Subunit of the CRISPR-Cas RNA Silencing ComplexOrigin of asymmetry in adenylyl cyclases: structures of Mycobacterium tuberculosis Rv1900cThe small molecule triclabendazole decreases the intracellular level of cyclic AMP and increases resistance to stress in Saccharomyces cerevisiaeAdenylate cyclase 1 (ADCY1) mutations cause recessive hearing impairment in humans and defects in hair cell function and hearing in zebrafish.The Concise Guide to PHARMACOLOGY 2013/14: enzymes.Structure-based development of novel adenylyl cyclase inhibitorsStructural and kinetic analyses of the interaction of anthrax adenylyl cyclase toxin with reaction products cAMP and pyrophosphate.Bis-halogen-anthraniloyl-substituted nucleoside 5'-triphosphates as potent and selective inhibitors of Bordetella pertussis adenylyl cyclase toxin.Inhibitors of membranous adenylyl cyclases.A conformational transition in the adenylyl cyclase catalytic site yields different binding modes for ribosyl-modified and unmodified nucleotide inhibitorsPhysiological roles for G protein-regulated adenylyl cyclase isoforms: insights from knockout and overexpression studies.Pharmacological distinction between soluble and transmembrane adenylyl cyclases.Catalytic Mechanism of Mammalian Adenylyl Cyclase: A Computational Investigation.Allosteric regulation of nucleotidyl cyclases: an emerging pharmacological target.A novel calcium-stimulated adenylyl cyclase from Trypanosoma cruzi, which interacts with the structural flagellar protein paraflagellar rod.The Molecular Pharmacology of G Protein Signaling Then and Now: A Tribute to Alfred G. Gilman.International Union of Basic and Clinical Pharmacology. CI. Structures and Small Molecule Modulators of Mammalian Adenylyl Cyclases.Gbetagamma activation site in adenylyl cyclase type II. Adenylyl cyclase type III is inhibited by Gbetagamma.Particulate adenylate cyclase plays a key role in human sperm olfactory receptor-mediated chemotaxis.Direct inhibition of type 5 adenylyl cyclase prevents myocardial apoptosis without functional deterioration.Differential inhibition of adenylyl cyclase isoforms and soluble guanylyl cyclase by purine and pyrimidine nucleotides.Mechanism of Galpha i-mediated inhibition of type V adenylyl cyclase.Differential inhibition of various adenylyl cyclase isoforms and soluble guanylyl cyclase by 2',3'-O-(2,4,6-trinitrophenyl)-substituted nucleoside 5'-triphosphatesType-specific regulation of adenylyl cyclase. Selective pharmacological stimulation and inhibition of adenylyl cyclase isoforms.Structure-based inhibitor discovery against adenylyl cyclase toxins from pathogenic bacteria that cause anthrax and whooping cough.Structural basis for the inhibition of mammalian membrane adenylyl cyclase by 2 '(3')-O-(N-Methylanthraniloyl)-guanosine 5 '-triphosphate.Role of the nucleotidyl cyclase helical domain in catalytically active dimer formation.Mammalian Nucleotidyl Cyclases and Their Nucleotide Binding Sites.Isolation, functional characterization, and transcriptome of Mastomys ileal enterochromaffin cells.Adenylate Cyclases of Trypanosoma brucei, Environmental Sensors and Controllers of Host Innate Immune Response.
P2860
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P2860
Molecular basis for P-site inhibition of adenylyl cyclase
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2000 nî lūn-bûn
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2000 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
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2000 թվականի նոյեմբերին հրատարակված գիտական հոդված
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2000年の論文
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2000年論文
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2000年論文
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2000年論文
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2000年論文
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2000年論文
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2000年论文
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name
Molecular basis for P-site inhibition of adenylyl cyclase
@ast
Molecular basis for P-site inhibition of adenylyl cyclase
@en
Molecular basis for P-site inhibition of adenylyl cyclase
@nl
type
label
Molecular basis for P-site inhibition of adenylyl cyclase
@ast
Molecular basis for P-site inhibition of adenylyl cyclase
@en
Molecular basis for P-site inhibition of adenylyl cyclase
@nl
prefLabel
Molecular basis for P-site inhibition of adenylyl cyclase
@ast
Molecular basis for P-site inhibition of adenylyl cyclase
@en
Molecular basis for P-site inhibition of adenylyl cyclase
@nl
P2093
P356
P1433
P1476
Molecular basis for P-site inhibition of adenylyl cyclase
@en
P2093
A G Gilman
C W Dessauer
L D Murray
R A Johnson
R K Sunahara
S R Sprang
P304
14464-14471
P356
10.1021/BI0015562
P407
P50
P577
2000-11-01T00:00:00Z