Population pharmacokinetic modelling of non-linear brain distribution of morphine: influence of active saturable influx and P-glycoprotein mediated efflux.
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P-glycoprotein modulates morphine uptake into the CNS: a role for the non-steroidal anti-inflammatory drug diclofenacChallenges of using in vitro data for modeling P-glycoprotein efflux in the blood-brain barrier.Enhanced analgesic responses after preferential delivery of morphine and fentanyl to the olfactory epithelium in rats.Kinetics of drug action in disease states: towards physiology-based pharmacodynamic (PBPD) models.Opioid analgesics and P-glycoprotein efflux transporters: a potential systems-level contribution to analgesic tolerance.The influence of age on the distribution of morphine and morphine-3-glucuronide across the blood-brain barrier in sheepEfflux transporters in the blood-brain interfaces--in vitro and in vivo methods and correlations.Transporter-Mediated Disposition of Opioids: Implications for Clinical Drug Interactions.A Generic Multi-Compartmental CNS Distribution Model Structure for 9 Drugs Allows Prediction of Human Brain Target Site ConcentrationsOpioids and the blood-brain barrier: a dynamic interaction with consequences on drug disposition in brain.Evidence of active transport involvement in morphine transport via MDCKII and MDCK-PGP cell lines.Impact of efflux transporters and of seizures on the pharmacokinetics of oxcarbazepine metabolite in the rat brain.Influence of biophase distribution and P-glycoprotein interaction on pharmacokinetic-pharmacodynamic modelling of the effects of morphine on the EEG.Pharmacokinetic modeling of non-linear brain distribution of fluvoxamine in the ratPredicting Drug Concentration-Time Profiles in Multiple CNS Compartments Using a Comprehensive Physiologically-Based Pharmacokinetic Model.Modelling the delay between pharmacokinetics and EEG effects of morphine in rats: binding kinetic versus effect compartment models
P2860
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P2860
Population pharmacokinetic modelling of non-linear brain distribution of morphine: influence of active saturable influx and P-glycoprotein mediated efflux.
description
2007 nî lūn-bûn
@nan
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
2007年论文
@zh
2007年论文
@zh-cn
name
Population pharmacokinetic mod ...... -glycoprotein mediated efflux.
@en
type
label
Population pharmacokinetic mod ...... -glycoprotein mediated efflux.
@en
prefLabel
Population pharmacokinetic mod ...... -glycoprotein mediated efflux.
@en
P2093
P2860
P356
P1476
Population pharmacokinetic mod ...... P-glycoprotein mediated efflux
@en
P2093
P2860
P304
P356
10.1038/SJ.BJP.0707257
P407
P577
2007-04-30T00:00:00Z