AM-411
AM-411 (part of the AM cannabinoid series) is an analgesic drug that is a cannabinoid agonist. It is a derivative of Δ8-THC substituted with an adamantyl group at the 3-position, demonstrating that the binding pocket for the alkyl chain at this position can accommodate significant bulk. AM-411 is a potent and fairly selective CB1 full agonist with a Ki of 6.80 nM, but is still also a moderately potent CB2 agonist with a Ki of 52.0 nM. It produces similar effects to other cannabinoid agonists such as analgesia, sedation, and anxiolysis.
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AM-411
AM-411 (part of the AM cannabinoid series) is an analgesic drug that is a cannabinoid agonist. It is a derivative of Δ8-THC substituted with an adamantyl group at the 3-position, demonstrating that the binding pocket for the alkyl chain at this position can accommodate significant bulk. AM-411 is a potent and fairly selective CB1 full agonist with a Ki of 6.80 nM, but is still also a moderately potent CB2 agonist with a Ki of 52.0 nM. It produces similar effects to other cannabinoid agonists such as analgesia, sedation, and anxiolysis.
has abstract
AM-411 (part of the AM cannabi ...... sia, sedation, and anxiolysis.
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CAS number
212835-02-4
ChEMBL
PubChem
Wikipage page ID
17,257,897
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Wikipage revision ID
1,022,956,999
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CAS number
ChEMBL
ChemSpiderID
IUPAC name
PubChem
SMILES
C5C6CC4CC5cccc1C2CC=CCC2C3C
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StdInChIKey
RPBMPWGKZFLMFN-OKFSJJLXSA-N
@en
verifiedrevid
415,995,491
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hypernym
comment
AM-411 (part of the AM cannabi ...... sia, sedation, and anxiolysis.
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label
AM-411
@en