4-Fluoropethidine
4-Fluoropethidine is a drug that is a derivative of pethidine (meperidine), which combines pethidine's opioid analgesic effects with increased monoamine reuptake inhibition. It is around 50% less potent than pethidine as an opioid analgesic, but conversely is 50% more potent as a dopamine reuptake inhibitor, with other derivatives such as the 4-iodo and 3,4-dichloro analogues being even more potent dopamine reuptake inhibitors again. However none of these compounds substitute for cocaine or produce stimulant effects in animals, suggesting that they still act primarily as opioid analgesic drugs in practice. Its action and degree of relation to pethidine means that it may be controlled in those countries which have laws about controlled-substance analogues; it is not itself listed in the Con
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4-Fluoropethidine
4-Fluoropethidine is a drug that is a derivative of pethidine (meperidine), which combines pethidine's opioid analgesic effects with increased monoamine reuptake inhibition. It is around 50% less potent than pethidine as an opioid analgesic, but conversely is 50% more potent as a dopamine reuptake inhibitor, with other derivatives such as the 4-iodo and 3,4-dichloro analogues being even more potent dopamine reuptake inhibitors again. However none of these compounds substitute for cocaine or produce stimulant effects in animals, suggesting that they still act primarily as opioid analgesic drugs in practice. Its action and degree of relation to pethidine means that it may be controlled in those countries which have laws about controlled-substance analogues; it is not itself listed in the Con
has abstract
4-Fluoropethidine is a drug th ...... ontrolled Substances Act 1970.
@en
ATC prefix
IUPAC name
ethyl 4-(4-fluorophenyl)-1-methylpiperidine-4-carboxylate
@en
PubChem
thumbnail
Wikipage page ID
27,972,299
Wikipage revision ID
720,786,834
ChEMBL
ChemSpiderID
molecular weight
2.65322e+2
smiles
StdInChIKey
CHOQGLPFQOQESN-UHFFFAOYSA-N
verifiedrevid
477,221,845
Watchedfields
subject
hypernym
comment
4-Fluoropethidine is a drug th ...... s not itself listed in the Con
@en
label
4-Fluoropethidine
@en