4-Phenylfentanyl
4-Phenylfentanyl is an opioid analgesic that is a derivative of fentanyl. It was developed during the course of research that ultimately resulted in super-potent opioid derivatives such as carfentanil, though it is a substantially less potent analogue. 4-Phenylfentanyl is around 8x the potency of fentanyl in analgesic tests on animals, but more complex 4-heteroaryl derivatives such as substituted thiophenes and thiazoles are more potent still, as they are closer bioisosteres to the 4-carbomethoxy group of carfentanil.
primaryTopic
4-Phenylfentanyl
4-Phenylfentanyl is an opioid analgesic that is a derivative of fentanyl. It was developed during the course of research that ultimately resulted in super-potent opioid derivatives such as carfentanil, though it is a substantially less potent analogue. 4-Phenylfentanyl is around 8x the potency of fentanyl in analgesic tests on animals, but more complex 4-heteroaryl derivatives such as substituted thiophenes and thiazoles are more potent still, as they are closer bioisosteres to the 4-carbomethoxy group of carfentanil.
has abstract
4-Phenylfentanyl is an opioid ...... erivatives continue to appear.
@en
ATC prefix
CAS number
120448-97-7
FDA UNII code
L9P31JAO37
IUPAC name
N-phenyl-N-[4-phenyl-1-(2-phenylethyl)piperidin-4-yl]propanamide
@en
PubChem
thumbnail
Wikipage page ID
27,961,855
Wikipage revision ID
727,673,759
ChemSpiderID
legal CA
legal UK
molecular weight
4.12566e+2
smiles
c3ccccc3CCNCCC2Nc4ccccc4
StdInChIKey
BXCJXJLHYMWMQU-UHFFFAOYSA-N
verifiedrevid
451,561,962
hypernym
comment
4-Phenylfentanyl is an opioid ...... omethoxy group of carfentanil.
@en
label
4-Phenylfentanyl
@en