Alphamethadol
Alphamethadol (INN), or α-methadol, also known as alfametadol, is a synthetic opioid analgesic. It is an isomer of dimepheptanol (methadol), the other being betamethadol (β-methadol). Alphamethadol is composed of two isomers itself, L-α-methadol, and D-α-methadol. The former compound, L-α-methadol, is an important active metabolite of levacetylmethadol (LAAM), an opioid substitute drug that is used clinically. Both of alphamethadol's isomers bind to and activate the μ-opioid receptor and are active as opioid analgesics, similarly to those of alphacetylmethadol (α-acetylmethadol).
primaryTopic
Alphamethadol
Alphamethadol (INN), or α-methadol, also known as alfametadol, is a synthetic opioid analgesic. It is an isomer of dimepheptanol (methadol), the other being betamethadol (β-methadol). Alphamethadol is composed of two isomers itself, L-α-methadol, and D-α-methadol. The former compound, L-α-methadol, is an important active metabolite of levacetylmethadol (LAAM), an opioid substitute drug that is used clinically. Both of alphamethadol's isomers bind to and activate the μ-opioid receptor and are active as opioid analgesics, similarly to those of alphacetylmethadol (α-acetylmethadol).
has abstract
Alfametadol – organiczny związ ...... ających z 1961 roku (wykaz I).
@pl
Alphamethadol (INN), or α-meth ...... ylmethadol (α-acetylmethadol).
@en
El alfametadol (α-metadol) es ...... es el betametadol (β-metadol).
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ATC prefix
CAS number
17199-54-1
IUPAC name
(3R,6R)-6-(dimethylamino)-4,4-diphenyl-3-heptanol
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PubChem
thumbnail
Wikipage page ID
14,743,728
Wikipage revision ID
721,307,216
ChEMBL
ChemSpiderID
legal CA
legal DE
legal US
molecular weight
3.11461e+2
smiles
StdInChIKey
QIRAYNIFEOXSPW-YLJYHZDGSA-N
comment
Alfametadol – organiczny związ ...... ających z 1961 roku (wykaz I).
@pl
Alphamethadol (INN), or α-meth ...... ylmethadol (α-acetylmethadol).
@en
El alfametadol (α-metadol) es ...... es el betametadol (β-metadol).
@es
label
Alfametadol
@es
Alfametadol
@pl
Alphamethadol
@en