Dissecting and designing inhibitor selectivity determinants at the S1 site using an artificial Ala190 protease (Ala190 uPA)
about
Allosteric antibody inhibition of human hepsin proteaseA urokinase-type plasminogen activator-inhibiting cyclic peptide with an unusual P2 residue and an extended protease binding surface demonstrates new modalities for enzyme inhibition.Cleavage specificity analysis of six type II transmembrane serine proteases (TTSPs) using PICS with proteome-derived peptide librariesThe cutting edge: membrane-anchored serine protease activities in the pericellular microenvironment.Design, synthesis and biological evaluation of PSMA/hepsin-targeted heterobivalent ligands.Expression, crystallization, and three-dimensional structure of the catalytic domain of human plasma kallikrein.Comparative binding energy analysis for binding affinity and target selectivity prediction.Mechanism-based selection of a potent kallikrein-related peptidase 7 inhibitor from a versatile library based on the sunflower trypsin inhibitor SFTI-1
P2860
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P2860
Dissecting and designing inhibitor selectivity determinants at the S1 site using an artificial Ala190 protease (Ala190 uPA)
description
2004 nî lūn-bûn
@nan
2004 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2004 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2004年の論文
@ja
2004年論文
@yue
2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
name
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@ast
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en-gb
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@nl
type
label
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@ast
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en-gb
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@nl
prefLabel
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@ast
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en-gb
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@nl
P2093
P1476
Dissecting and designing inhib ...... l Ala190 protease (Ala190 uPA)
@en
P2093
Bradley A Katz
Christine Luong
Erik Gjerstad
Erik Verner
James W Janc
John R Somoza
Joseph D Ho
Kyle Mortara
P304
P356
10.1016/J.JMB.2004.09.032
P407
P577
2004-11-19T00:00:00Z