A new class of symmetric bisbenzimidazole-based DNA minor groove-binding agents showing antitumor activity
about
The discovery of a novel antibiotic for the treatment of Clostridium difficile infections: a story of an effective academic–industrial partnershipSTK295900, a dual inhibitor of topoisomerase 1 and 2, induces G(2) arrest in the absence of DNA damage.Growth Inhibitory Activity of a Bis-benzimidazole-Bridged Arene Ruthenium Metalla-Rectangle and Prism.Sequence-specific minor groove binding by bis-benzimidazoles: water molecules in ligand recognition.A Personal History of Quadruplex-Small Molecule Targeting.Synthesis and biological evaluation of benzimidazole-linked 1,2,3-triazole congeners as agentsFacile and efficient one-pot synthesis of benzimidazoles using lanthanum chlorideUse of the in vivo hollow fiber assay in natural products anticancer drug discovery.Minor grove binding ligands disrupt PARP-1 activation pathways.New Route Synthesis of Thiadiazoles, Bisthiadiazoles, Thiadiazolotriazines, and Pyrazolothiadiazoles Based on Hydrazonoyl Halides and Dihydrazinylthiadiazole.Bis(1-benzyl-1H-benzimidazole-κN (3))di-chlorido-zincZinc(II) complexes containing bis-benzimidazole derivatives as a new class of apoptosis inducers that trigger DNA damage-mediated p53 phosphorylation in cancer cells.Synthesis and anticancer activity evaluation of N-[4-(2-methylthiazol-4-yl)phenyl]acetamide derivatives containing (benz)azole moiety.Ruthenium complexes containing 2,6-bis(benzimidazolyl)pyridine derivatives induce cancer cell apoptosis by triggering DNA damage-mediated p53 phosphorylation.Synthesis and characterization of the ligand based on benzimidazole and its copper complex: DNA binding and antioxidant activity.Synthesis, biological evaluation, and modeling of dimeric PPI analogues as novel DNA minor groove binders.Synthesis of diphenylcarbazoles as cytotoxic DNA binding agents.Graph theoretical analysis, insilico modeling, design, and synthesis of compounds containing benzimidazole skeleton as antidepressant agents.Di- and triheteroarylalkanes via self-condensation and intramolecular Friedel-Crafts type reaction of heteroaryl alcohols.Synthesis, Characterization, and Application of Poly(N,N′-dibromo-N-ethylnaphthyl-2,7-disulfonamide) as an Efficient Reagent for the Synthesis of 2-Arylbenzimidazole and 2-Aryl-1-arylmethyl-1H-1,3-benzimidazole DerivativesRemarkable Acceleration of Benzimidazole Synthesis and Cyanosilylation Reactions in a Supramolecular Solid Catalyst
P2860
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P2860
A new class of symmetric bisbenzimidazole-based DNA minor groove-binding agents showing antitumor activity
description
2001 nî lūn-bûn
@nan
2001 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2001 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2001年の論文
@ja
2001年論文
@yue
2001年論文
@zh-hant
2001年論文
@zh-hk
2001年論文
@zh-mo
2001年論文
@zh-tw
2001年论文
@wuu
name
A new class of symmetric bisbe ...... nts showing antitumor activity
@ast
A new class of symmetric bisbe ...... nts showing antitumor activity
@en
A new class of symmetric bisbe ...... nts showing antitumor activity
@nl
type
label
A new class of symmetric bisbe ...... nts showing antitumor activity
@ast
A new class of symmetric bisbe ...... nts showing antitumor activity
@en
A new class of symmetric bisbe ...... nts showing antitumor activity
@nl
prefLabel
A new class of symmetric bisbe ...... nts showing antitumor activity
@ast
A new class of symmetric bisbe ...... nts showing antitumor activity
@en
A new class of symmetric bisbe ...... nts showing antitumor activity
@nl
P2093
P356
P1476
A new class of symmetric bisbe ...... nts showing antitumor activity
@en
P2093
E Johansson
G Parkinson
L R Kelland
Y Opoku-Boahen
P304
P356
10.1021/JM000297B
P407
P577
2001-01-18T00:00:00Z