Huprine derivatives as sub-nanomolar human acetylcholinesterase inhibitors: from rational design to validation by X-ray crystallography

Huprine derivatives as sub-nanomolar human acetylcholinesterase inhibitors: from rational design to validation by X-ray crystallography

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http://www.wikidata.org/entity/Q27675368
Human butyrylcholinesterase produced in insect cells: huprine-based affinity purification and crystal structureCrystal structures of human cholinesterases in complex with huprine W and tacrine: elements of specificity for anti-Alzheimer's drugs targeting acetyl- and butyryl-cholinesteraseCorrelation of the dynamics of native human acetylcholinesterase and its inhibited huperzine A counterpart from sub-picoseconds to nanoseconds.New insights into the kinetic target-guided synthesis of protein ligands.Recent developments in structural studies on acetylcholinesterase.Reaction site-driven regioselective synthesis of AChE inhibitors.Comparison of the Binding of Reversible Inhibitors to Human Butyrylcholinesterase and Acetylcholinesterase: A Crystallographic, Kinetic and Calorimetric Study.A selective and sensitive near-infrared fluorescent probe for acetylcholinesterase imaging.5-Methyl--(8-(5,6,7,8-tetrahydroacridin-9-ylamino)octyl)-5-indolo[2,3-]quinolin-11-amine: a highly potent human cholinesterase inhibitor
P2860

Huprine derivatives as sub-nanomolar human acetylcholinesterase inhibitors: from rational design to validation by X-ray crystallography

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http://www.wikidata.org/entity/Q27675368
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2012 nî lūn-bûn
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2012 թուականի Մարտին հրատարակուած գիտական յօդուած
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2012 թվականի մարտին հրատարակված գիտական հոդված
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2012年の論文
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2012年論文
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2012年論文
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2012年論文
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2012年論文
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2012年論文
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2012年论文
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Huprine derivatives as sub-nan ...... ation by X-ray crystallography
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Huprine derivatives as sub-nan ...... ation by X-ray crystallography
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Huprine derivatives as sub-nan ...... ation by X-ray crystallography
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type
label
Huprine derivatives as sub-nan ...... ation by X-ray crystallography
@ast
Huprine derivatives as sub-nan ...... ation by X-ray crystallography
@en
Huprine derivatives as sub-nan ...... ation by X-ray crystallography
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prefLabel
Huprine derivatives as sub-nan ...... ation by X-ray crystallography
@ast
Huprine derivatives as sub-nan ...... ation by X-ray crystallography
@en
Huprine derivatives as sub-nan ...... ation by X-ray crystallography
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Huprine derivatives as sub-nan ...... ation by X-ray crystallography
@en
P2093
P2860
P304
P31
P356
P433
P478
P50
P577
P5875
P698
P921