Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds
about
Crystal structure of human CK2α at 1.06 Å resolutionPharmacophore modeling and in silico toxicity assessment of potential anticancer agents from African medicinal plantsPhosphoproteomics Identifies CK2 as a Negative Regulator of Beige Adipocyte Thermogenesis and Energy Expenditure.Exploring the prominent performance of CX-4945 derivatives as protein kinase CK2 inhibitors by a combined computational study.Identification of potential CCR5 inhibitors through pharmacophore-based virtual screening, molecular dynamics simulation and binding free energy analysis.Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles.A Selective Biligand Inhibitor of CK2 Increases Caspase-3 Activity in Cancer Cells and Inhibits Platelet Aggregation.Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors.
P2860
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P2860
Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds
description
2012 nî lūn-bûn
@nan
2012 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի մարտին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@ast
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@en
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@nl
type
label
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@ast
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@en
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@nl
prefLabel
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@ast
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@en
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@nl
P2093
P3181
P356
P1476
Structure-based design of nove ...... rs with phenyl-azole scaffolds
@en
P2093
Akira Hirasawa
Gozoh Tsujimoto
Hiroaki Ohno
Isao Nakanishi
Katsumi Murata
Kazuo Kitaura
Misato Yasue
Nobutaka Fujii
Ryosuke Misu
Shinya Nakamura
P304
P3181
P356
10.1021/JM2015167
P407
P577
2012-03-22T00:00:00Z