Synthesis and structure-activity relationships for 1-(4-(piperidin-1-ylsulfonyl)phenyl)pyrrolidin-2-ones as novel non-carboxylate inhibitors of the aldo-keto reductase enzyme AKR1C3

Synthesis and structure-activity relationships for 1-(4-(piperidin-1-ylsulfonyl)phenyl)pyrrolidin-2-ones as novel non-carboxylate inhibitors of the aldo-keto reductase enzyme AKR1C3

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http://www.wikidata.org/entity/Q27684103
Structures of complexes of type 5 17β-hydroxysteroid dehydrogenase with structurally diverse inhibitors: insights into the conformational changes upon inhibitor bindingThe Activity of SN33638, an Inhibitor of AKR1C3, on Testosterone and 17β-Estradiol Production and Function in Castration-Resistant Prostate Cancer and ER-Positive Breast Cancer.Screening baccharin analogs as selective inhibitors against type 5 17β-hydroxysteroid dehydrogenase (AKR1C3).Aldo-Keto Reductase AKR1C1-AKR1C4: Functions, Regulation, and Intervention for Anti-cancer Therapy.Discovery of (R)-2-(6-Methoxynaphthalen-2-yl)butanoic Acid as a Potent and Selective Aldo-keto Reductase 1C3 Inhibitor.AKR1C3 Inhibition Therapy in Castration-Resistant Prostate Cancer and Breast Cancer: Lessons from Responses to SN33638.Aldo-Keto Reductase (AKR) 1C3 inhibitors: a patent review.Synthesis and molecular docking studies of some 4-phthalimidobenzenesulfonamide derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors.
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Synthesis and structure-activity relationships for 1-(4-(piperidin-1-ylsulfonyl)phenyl)pyrrolidin-2-ones as novel non-carboxylate inhibitors of the aldo-keto reductase enzyme AKR1C3

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http://www.wikidata.org/entity/Q27684103
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2013 nî lūn-bûn
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2013 թուականի Ապրիլին հրատարակուած գիտական յօդուած
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2013 թվականի ապրիլին հրատարակված գիտական հոդված
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2013年の論文
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2013年学术文章
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2013年学术文章
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2013年学术文章
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2013年学术文章
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2013年學術文章
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Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@ast
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@en
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@nl
type
label
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@ast
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@en
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@nl
prefLabel
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@ast
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@en
Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@nl
P1433
P1476
P2093
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P356
P478
P50
P577
P698
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Synthesis and structure-activi ...... o-keto reductase enzyme AKR1C3
@en
P2093
P304
P31
P356
10.1016/J.EJMECH.2013.01.047
P478
P50
P577
P698