Discovery of 1H-pyrazol-3(2H)-ones as potent and selective inhibitors of protein kinase R-like endoplasmic reticulum kinase (PERK)
about
Elucidation of molecular mechanism of stability of the heme-regulated eIF2α kinase upon binding of its ligand, hemin in its catalytic kinase domain.Protein kinase R(PKR)-like endoplasmic reticulum kinase (PERK) inhibitors: a patent review (2010-2015).The entangled ER-mitochondrial axis as a potential therapeutic strategy in neurodegeneration: A tangled duo unchained.Endoplasmic Reticulum Stress Sensor IRE1α Enhances IL-23 Expression by Human Dendritic Cells.The eIF2-alpha kinase HRI: a potential target beyond the red blood cell.A facile and general acid-catalyzed deuteration at methyl groups of N-heteroarylmethanes.When PERK inhibitors turn out to be new potent RIPK1 inhibitors: critical issues on the specificity and use of GSK2606414 and GSK2656157.PERK signalling pathway mediates single prolonged stress-induced dysfunction of medial prefrontal cortex neurons.Triazolo[4,5]pyrimidines as Validated General Control Nonderepressible 2 (GCN2) Protein Kinase Inhibitors Reduce Growth of Leukemia Cells
P2860
Q38621770-122869E3-4FFA-4554-AC9E-AA33D81812ECQ38819666-084AD62C-59D2-4207-9BA7-0663794F2422Q38841508-3176C05E-4502-4627-9548-3B6C4931D043Q41102193-E700D672-B8C4-4997-940A-70C0588932C7Q47611637-B1CFFFD7-0837-4F40-A854-A485F9D7A98AQ48156317-A18A253D-D11D-4D0B-BC78-888DD79549A2Q49099457-5A8DE2F1-3026-4E37-ABFA-B503B2236DC1Q50445421-F74C3F92-1E82-4E0A-A752-42B53B03173FQ58547957-9E58C067-9539-4C77-85FA-7A573EC84A31
P2860
Discovery of 1H-pyrazol-3(2H)-ones as potent and selective inhibitors of protein kinase R-like endoplasmic reticulum kinase (PERK)
description
2015 nî lūn-bûn
@nan
2015 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2015 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
name
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@ast
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@en
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@nl
type
label
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@ast
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@en
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@nl
prefLabel
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@ast
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@en
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@nl
P2093
P356
P1476
Discovery of 1H-pyrazol-3(2H)- ...... lasmic reticulum kinase (PERK)
@en
P2093
Adrian L Smith
Alexander M Long
David Powers
Holger Beckmann
J Russell Lipford
Jennifer Dao
Katja Labitzke
Kenneth R Dellamaggiore
Kristin L Andrews
P304
P356
10.1021/JM5017494
P407
P577
2015-02-12T00:00:00Z