Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH 17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor RORγ
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Fragment Screening of RORγt Using Cocktail Crystallography: Identification of Simultaneous Binding of Multiple FragmentsN-Arylsulfonyl Indolines as Retinoic Acid Receptor-Related Orphan Receptor γ (RORγ) Agonists.Modular Bi-Directional One-Pot Strategies for the Diastereoselective Synthesis of Structurally Diverse Collections of Constrained β-Carboline-Benzoxazepines.Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.Structural States of RORγt: X-ray Elucidation of Molecular Mechanisms and Binding Interactions for Natural and Synthetic Compounds.Ternary complex of human RORγ ligand-binding domain, inverse agonist and SMRT peptide shows a unique mechanism of corepressor recruitment.
P2860
Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH 17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor RORγ
description
2016 nî lūn-bûn
@nan
2016 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2016 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@ast
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@en
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@nl
type
label
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@ast
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@en
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@nl
prefLabel
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@ast
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@en
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@nl
P2093
P2860
P356
P1433
P1476
Benzoxazepines Achieve Potent ...... e to the Nuclear Receptor RORγ
@en
P2093
Agnes Leffler
Anna Aagaard
Eva L Hansson
Hanna Grindebacke
Hongbin Ge
Jane McPheat
Jenny Bernström
Johan Jirholt
Pia Hansson
Roine I Olsson
P2860
P304
P356
10.1002/CMDC.201500432
P50
P577
2015-11-10T00:00:00Z