Important Hydrogen Bond Networks in Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Design Revealed by Crystal Structures of Imidazoleisoindole Derivatives with IDO1
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Erylusamides: Novel Atypical Glycolipids from Erylus cf. deficiensStructural Study of a Flexible Active Site Loop in Human Indoleamine 2,3-Dioxygenase and Its Functional Implications.Discovery of a Novel Scaffold as an Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Based on the Pyrrolopiperazinone Alkaloid, Longamide B.Distinct roles of immunoreceptor tyrosine-based motifs in immunosuppressive indoleamine 2,3-dioxygenase 1.In silico discovery and therapeutic potential of IDO1 and TDO2 inhibitors.Binding properties of different categories of IDO1 inhibitors: a microscale thermophoresis study.Major developments in the design of inhibitors along the kynurenine pathway.Abnormal kynurenine pathway of tryptophan catabolism in cardiovascular diseases.Heme-containing enzymes and inhibitors for tryptophan metabolism.Evaluation of radiofluorinated carboximidamides as potential IDO-targeted PET tracers for cancer imaging.A short history of heme dioxygenases: rise, fall and rise again.Structural insights into substrate and inhibitor binding sites in human indoleamine 2,3-dioxygenase 1.Discovery of IDO1 Inhibitors: From Bench to Bedside.Synthesis and Molecular Modeling Studies of N'-Hydroxyindazolecarboximidamides as Novel Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors.Different Mechanisms of Catalytic Complex Formation in Two L-Tryptophan Processing Dioxygenases.Identification of Potent Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors Based on a Phenylimidazole Scaffold.Inflammatory Reprogramming with IDO1 Inhibitors: Turning Immunologically Unresponsive 'Cold' Tumors 'Hot'.Discovery of Novel Inhibitors of Indoleamine 2,3-Dioxygenase 1 Through Structure-Based Virtual Screening.Insights into the mechanism of inhibition of tryptophan 2,3-dioxygenase by isatin derivatives.
P2860
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P2860
Important Hydrogen Bond Networks in Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Design Revealed by Crystal Structures of Imidazoleisoindole Derivatives with IDO1
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2016 nî lūn-bûn
@nan
2016 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2016 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@ast
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@en
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@nl
type
label
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@ast
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@en
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@nl
prefLabel
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@ast
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@en
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@nl
P2093
P3181
P1476
Important Hydrogen Bond Networ ...... soindole Derivatives with IDO1
@en
P2093
Chen-Tso Tseng
Chia-Yi Cheng
Chih-Hsiang Tu
Ching-Cheng Hsueh
Chuan Shih
Fang-Yu Liao
Jen-Shin Song
Jian-Sung Wu
Kak-Shan Shia
Lung-Chun Lee
P304
P3181
P356
10.1021/ACS.JMEDCHEM.5B01390
P407
P577
2016-01-14T00:00:00Z