Qualitative and quantitative assessment of relative agonist efficacy
about
Molecular mechanisms of action and in vivo validation of an M4 muscarinic acetylcholine receptor allosteric modulator with potential antipsychotic propertiesFrom 'captive' agonism to insurmountable antagonism: demonstrating the power of analytical pharmacology.Isolation and pharmacological characterization of AdTx1, a natural peptide displaying specific insurmountable antagonism of the alpha1A-adrenoceptor.μ-opioid receptors: correlation of agonist efficacy for signalling with ability to activate internalization.Mu-opioid receptor desensitization: is morphine different?Ligand bias at the μ-opioid receptor.Efficacy and ligand bias at the μ-opioid receptor.Superagonism at G protein-coupled receptors and beyond.Characterization of a Novel M1 Muscarinic Acetylcholine Receptor Positive Allosteric Modulator Radioligand, [3H]PT-1284.A novel mechanism of G protein-coupled receptor functional selectivity. Muscarinic partial agonist McN-A-343 as a bitopic orthosteric/allosteric ligand.Measurement of smooth muscle function in the isolated tissue bath-applications to pharmacology research.Agonist stimulation at human μ opioid receptors in a [(35)S]GTPγS incorporation assay: observation of "bell-shaped" concentration-response relationships under conditions of strong receptor G protein coupling.Multiple Routes to Oestrogen Antagonism.
P2860
Q30498538-FD1798B9-DCBF-48C8-B079-F717B452A564Q32115544-C25B68E5-D456-4D5A-B971-88EC528817E4Q33673036-2FFBEC2A-2B9D-41ED-B89A-D4EF1A1F356FQ34310081-B4CD2204-5D66-4EDC-A05F-11551EC4DBADQ35927616-F2549530-2567-4B9B-A723-067FA69D788FQ38077231-23B70F96-33DA-465E-AF97-29DDAFC9D6DBQ38104365-3DCAA9B5-1EC6-41B7-B88D-9AAB469BE0A1Q38567235-6E3149C8-CF97-4951-9DD4-E53FBB143256Q38759673-A9545D6F-37A7-4DA9-8007-B5C34C9D3239Q39947679-E004C7FE-8E48-4226-98F0-D19DFFAB1BE3Q40254846-0CDB05F9-B53F-40C0-86AD-384B20CE26D0Q42483748-69630093-D97E-4407-BC7E-277B2D68955DQ55452150-9FC8ED35-06A6-4AEE-950F-3445E1C00BE0
P2860
Qualitative and quantitative assessment of relative agonist efficacy
description
1999 nî lūn-bûn
@nan
1999 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
Qualitative and quantitative assessment of relative agonist efficacy
@ast
Qualitative and quantitative assessment of relative agonist efficacy
@en
Qualitative and quantitative assessment of relative agonist efficacy
@nl
type
label
Qualitative and quantitative assessment of relative agonist efficacy
@ast
Qualitative and quantitative assessment of relative agonist efficacy
@en
Qualitative and quantitative assessment of relative agonist efficacy
@nl
prefLabel
Qualitative and quantitative assessment of relative agonist efficacy
@ast
Qualitative and quantitative assessment of relative agonist efficacy
@en
Qualitative and quantitative assessment of relative agonist efficacy
@nl
P1476
Qualitative and quantitative assessment of relative agonist efficacy
@en
P2093
A Christopoulos
E E El-Fakahany
P304
P356
10.1016/S0006-2952(99)00087-8
P407
P577
1999-09-01T00:00:00Z