Design, synthesis, structure-activity relationship, and in vivo activity of azabicyclic aryl amides as alpha7 nicotinic acetylcholine receptor agonists
about
Nicotine decreases DNA methyltransferase 1 expression and glutamic acid decarboxylase 67 promoter methylation in GABAergic interneuronsCreating an 7 Nicotinic Acetylcholine Recognition Domain from the Acetylcholine-binding Protein: CRYSTALLOGRAPHIC AND LIGAND SELECTIVITY ANALYSESExploring chemical space for drug discovery using the chemical universe database.High throughput electrophysiology with Xenopus oocytesAlpha7 nicotinic acetylcholine receptor: a link between inflammation and neurodegeneration.Chemical and genetic engineering of selective ion channel-ligand interactionsα7 Nicotinic Receptor Agonists: Potential Therapeutic Drugs for Treatment of Cognitive Impairments in Schizophrenia and Alzheimer's Disease.Evidence of BrdU-positive retinal neurons after application of an Alpha7 nicotinic acetylcholine receptor agonist.Preclinical characterization of A-582941: a novel alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties.Exploring α7-Nicotinic Receptor Ligand Diversity by Scaffold Enumeration from the Chemical Universe Database GDBRetinal ganglion cell neuroprotection induced by activation of alpha7 nicotinic acetylcholine receptors.Contribution of α7 nicotinic receptor to airway epithelium dysfunction under nicotine exposureReducing inflammation and rescuing FTD-related behavioral deficits in progranulin-deficient mice with α7 nicotinic acetylcholine receptor agonistsRecent advances in the development of novel pharmacological agents for the treatment of cognitive impairments in schizophrenia.Targeting of α7 Nicotinic Acetylcholine Receptors in the Treatment of Schizophrenia and the Use of Auditory Sensory Gating as a Translational BiomarkerAlpha7 neuronal nicotinic receptors as a drug target in schizophrenia.The therapeutic potential of α7 nicotinic acetylcholine receptor (α7 nAChR) agonists for the treatment of the cognitive deficits associated with schizophrenia.α7 nicotinic acetylcholine receptor agonist PNU-282987 attenuates early brain injury in a perforation model of subarachnoid hemorrhage in rats.Activation of Alpha-7 Nicotinic Acetylcholine Receptor Reduces Brain Edema in Mice with Ischemic Stroke and Bone Fracture.The nicotinic acetylcholine receptor as a target for antidepressant drug development.Preclinical Characterization of A-582941: A Novel α7 Neuronal Nicotinic Receptor Agonist with Broad Spectrum Cognition-Enhancing Properties
P2860
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P2860
Design, synthesis, structure-activity relationship, and in vivo activity of azabicyclic aryl amides as alpha7 nicotinic acetylcholine receptor agonists
description
2006 nî lūn-bûn
@nan
2006 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2006 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
name
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@ast
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@en
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@nl
type
label
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@ast
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@en
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@nl
prefLabel
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@ast
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@en
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@nl
P2093
P1476
Design, synthesis, structure-a ...... cetylcholine receptor agonists
@en
P2093
Barbara A Olson
Brad A Acker
Brandon J Margolis
Brian A Staton
Bruce A Thornburgh
Bruce N Rogers
Daniel P Walker
David W Piotrowski
Donn G Wishka
E Jon Jacobsen
P304
P356
10.1016/J.BMC.2006.09.019
P407
P577
2006-12-15T00:00:00Z