1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist

1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist

Item
http://www.wikidata.org/entity/Q28283767
In silico molecular comparisons of C. elegans and mammalian pharmacology identify distinct targets that regulate feedingCharacterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonistOxytocin signaling in mouse taste budsOxytocin and vasopressin agonists and antagonists as research tools and potential therapeutics.REVIEW: Oxytocin: Crossing the bridge between basic science and pharmacotherapyA Gly/Ala switch contributes to high affinity binding of benzoxazinone-based non-peptide oxytocin receptor antagonists.Pharmacologic characterization of the oxytocin receptor in human uterine smooth muscle cells.Selectivity of d[Cha4]AVP and SSR149415 at human vasopressin and oxytocin receptors: evidence that SSR149415 is a mixed vasopressin V1b/oxytocin receptor antagonistSynthesis and evaluation of C-11, F-18 and I-125 small molecule radioligands for detecting oxytocin receptors.Differential contributions of vasopressin V1A and oxytocin receptors in the amygdala to pain-related behaviors in rats.Modeling the human oxytocin receptor for drug discovery efforts.Small molecule ligands for oxytocin and vasopressin receptors.Identification of an extracellular segment of the oxytocin receptor providing agonist-specific binding epitopes.Design of oxytocin antagonists, which are more selective than atosiban.
P2860

1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist

Item
http://www.wikidata.org/entity/Q28283767
description
1995 nî lūn-bûn
@nan
1995 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
1995 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
name
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@ast
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@en
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@nl
type
label
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@ast
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@en
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@nl
prefLabel
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@ast
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@en
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@nl
P1433
P1476
P2093
P304
P31
P356
P407
P433
P478
P577
P698
P921
P356
P1433
P1476
1-(1-[4-[(N-acetyl-4-piperidin ...... on-peptide oxytocin antagonist
@en
P2093
P304
P31
P356
P407
P433
P478
P577
P698
P921