Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
about
Principles of agonist recognition in Cys-loop receptorsAllosteric activation mechanism of the cys-loop receptorsBinding of muscimol-conjugated quantum dots to GABAC receptors.A residue in loop 9 of the beta2-subunit stabilizes the closed state of the GABAA receptor.Ligand- and subunit-specific conformational changes in the ligand-binding domain and the TM2-TM3 linker of {alpha}1 {beta}2 {gamma}2 GABAA receptorsGABA signalling modulates plant growth by directly regulating the activity of plant-specific anion transportersAllosteric modulation of retinal GABA receptors by ascorbic acid.2-Aminoethyl methylphosphonate, a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors.Functional Impact of 14 Single Nucleotide Polymorphisms Causing Missense Mutations of Human α7 Nicotinic Receptor.Molecular cloning and expression of a GABA receptor subunit from the crayfish Procambarus clarkii.Structurally diverse GABA antagonists interact differently with open and closed conformational states of the ρ1 receptor.Nitric oxide potentiation of the homomeric ρ1 GABA(C) receptor function.Quantum dot conjugates of GABA and muscimol: binding to α1β2γ2 and ρ1 GABA(A) receptors.Structural rearrangements in loop F of the GABA receptor signal ligand binding, not channel activation.Structural model of rho1 GABAC receptor based on evolutionary analysis: Testing of predicted protein-protein interactions involved in receptor assembly and function.The role of Loop F in the activation of the GABA receptor.An intracellular redox sensor for reactive oxygen species at the M3-M4 linker of GABAA ρ1 receptors.The structural basis of function in Cys-loop receptors.An Update on GABAρ Receptors.Synaptic neurotransmitter-gated receptorsCysteine modification reveals which subunits form the ligand binding site in human heteromeric 5-HT3AB receptors.GABA-ρ receptors: distinctive functions and molecular pharmacology.A hydrophobic area of the GABA ρ₁ receptor containing phenylalanine 124 influences both receptor activation and deactivation.Locating the carboxylate group of GABA in the homomeric rho GABA(A) receptor ligand-binding pocket.Mutagenesis and molecular modeling reveal the importance of the 5-HT3 receptor F-loop.Molecular dynamics simulations of GABA binding to the GABAC receptor: the role of Arg104.Unbinding pathways of an agonist and an antagonist from the 5-HT3 receptorAgonist- and antagonist-induced conformational changes of loop F and their contributions to the rho1 GABA receptor function.Redox modulation of homomeric rho1 GABA receptors.Antagonistic effect of dopamine structural analogues on human GABAρ1 receptor.Negative modulation of the GABAA ρ1 receptor function by l-cysteine.Discovery of α-Substituted Imidazole-4-acetic Acid Analogues as a Novel Class of ρ1 γ-Aminobutyric Acid Type A Receptor Antagonists with Effect on Retinal Vascular Tone.
P2860
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P2860
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
description
2005 nî lūn-bûn
@nan
2005 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2005年の論文
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2005年学术文章
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2005年学术文章
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2005年学术文章
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2005年学术文章
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2005年学术文章
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2005年學術文章
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name
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@ast
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@en
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@nl
type
label
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@ast
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@en
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@nl
prefLabel
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@ast
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@en
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@nl
P2093
P2860
P356
P1476
Mapping the rho1 GABA(C) receptor agonist binding pocket. Constructing a complete model
@en
P2093
Anna Sedelnikova
Craig D Smith
David S Weiss
Delores Davis
Stanislav O Zakharkin
Yongchang Chang
P2860
P304
P356
10.1074/JBC.M409908200
P407
P577
2005-01-14T00:00:00Z