Synthesis, dopamine transporter affinity, dopamine uptake inhibition, and locomotor stimulant activity of 2-substituted 3 beta-phenyltropane derivatives
about
Development of 3-phenyltropane analogues with high affinity for the dopamine and serotonin transporters and low affinity for the norepinephrine transporter.Probes for the dopamine transporter: new leads toward a cocaine-abuse therapeutic--A focus on analogues of benztropine and rimcazole.Low and high affinity dopamine transporter inhibitors block dopamine uptake within 5 sec of intravenous injection.Synthesis and structure-activity relationship of 3beta-(4-alkylthio, -methylsulfinyl, and -methylsulfonylphenyl)tropane and 3beta-(4-alkylthiophenyl)nortropane derivatives for monoamine transporters.Synthesis and receptor binding properties of 2beta-alkynyl and 2beta-(1,2,3-triazol)substituted 3beta-(substituted phenyl)tropane derivatives.Synthesis and monoamine transporter binding properties of 2beta-[3'-(substituted benzyl)isoxazol-5-yl]- and 2beta-[3'-methyl-4'-(substituted phenyl)isoxazol-5-yl]-3beta-(substituted phenyl)tropanes.
P2860
Synthesis, dopamine transporter affinity, dopamine uptake inhibition, and locomotor stimulant activity of 2-substituted 3 beta-phenyltropane derivatives
description
1997 nî lūn-bûn
@nan
1997 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
1997 թվականի մարտին հրատարակված գիտական հոդված
@hy
1997年の論文
@ja
1997年論文
@yue
1997年論文
@zh-hant
1997年論文
@zh-hk
1997年論文
@zh-mo
1997年論文
@zh-tw
1997年论文
@wuu
name
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@ast
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@en
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@nl
type
label
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@ast
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@en
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@nl
prefLabel
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@ast
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@en
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@nl
P2093
P356
P1476
Synthesis, dopamine transporte ...... beta-phenyltropane derivatives
@en
P2093
P304
P356
10.1021/JM960739C
P407
P577
1997-03-01T00:00:00Z