Relationships between inhibition constants, inhibitor concentrations for 50% inhibition and types of inhibition: new ways of analysing data
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Mode of Action, In Vitro Activity, and In Vivo Efficacy of AFN-1252, a Selective Antistaphylococcal FabI InhibitorKinetic studies of rat liver hexokinase D ('glucokinase') in non-co-operative conditions show an ordered mechanism with MgADP as the last product to be releasedActive-learning exercises to teach drug-receptor interactions in a medicinal chemistry courseLog-scale dose response of inhibitors on a chip.Inhibitors of the mitochondrial citrate transport protein: validation of the role of substrate binding residues and discovery of the first purely competitive inhibitor.Zinc-binding groups modulate selective inhibition of MMPs.Cysteine residues 244 and 458-459 within the catalytic subunit of Na,K-ATPase control the enzyme's hydrolytic and signaling function under hypoxic conditions.Multi-target QSAR modelling in the analysis and design of HIV-HCV co-inhibitors: an in-silico study.Intracellular function of interleukin-1 receptor antagonist in ischemic cardiomyocytes.FTY720 analogues as sphingosine kinase 1 inhibitors: enzyme inhibition kinetics, allosterism, proteasomal degradation, and actin rearrangement in MCF-7 breast cancer cells.Inhibition of secreted phospholipase A2 by neuron survival and anti-inflammatory peptide CHEC-9(R)-FTY720 methyl ether is a specific sphingosine kinase 2 inhibitor: Effect on sphingosine kinase 2 expression in HEK 293 cells and actin rearrangement and survival of MCF-7 breast cancer cells.Inhibitors of the AAA+ chaperone p97S-glutathionylation of the Na,K-ATPase catalytic α subunit is a determinant of the enzyme redox sensitivityOxygen-induced Regulation of Na/K ATPase in cerebellar granule cellsBone sialoprotein binding to matrix metalloproteinase-2 alters enzyme inhibition kinetics.Caffeine inhibits acetylcholinesterase, but not butyrylcholinesteraseSubstituted hippurates and hippurate analogs as substrates and inhibitors of peptidylglycine alpha-hydroxylating monooxygenase (PHM).Characterizing metabolic inhibition using electrochemical enzyme/DNA biosensorsThe yeast mitochondrial citrate transport protein: identification of the Lysine residues responsible for inhibition mediated by Pyridoxal 5'-phosphate.Binding of hematin by a new class of glutathione transferase from the blood-feeding parasitic nematode Haemonchus contortus.Determination of half-maximal inhibitory concentration using biosensor-based protein interaction analysis.Resveratrol dimers are novel sphingosine kinase 1 inhibitors and affect sphingosine kinase 1 expression and cancer cell growth and survivalUnified Modeling of Familial Mediterranean Fever and Cryopyrin Associated Periodic Syndromes.External mechanical force as an inhibition process in kinesin's motion.Overexpression of wild-type aspartokinase increases L-lysine production in the thermotolerant methylotrophic bacterium Bacillus methanolicus.Ligand binding phenomena that pertain to the metabolic function of renalase.An automated framework for QSAR model building.Synthesis and structure-activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis
P2860
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P2860
Relationships between inhibition constants, inhibitor concentrations for 50% inhibition and types of inhibition: new ways of analysing data
description
2001 nî lūn-bûn
@nan
2001 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2001 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2001年の論文
@ja
2001年論文
@yue
2001年論文
@zh-hant
2001年論文
@zh-hk
2001年論文
@zh-mo
2001年論文
@zh-tw
2001年论文
@wuu
name
Relationships between inhibiti ...... on: new ways of analysing data
@ast
Relationships between inhibiti ...... on: new ways of analysing data
@en
Relationships between inhibiti ...... on: new ways of analysing data
@nl
type
label
Relationships between inhibiti ...... on: new ways of analysing data
@ast
Relationships between inhibiti ...... on: new ways of analysing data
@en
Relationships between inhibiti ...... on: new ways of analysing data
@nl
prefLabel
Relationships between inhibiti ...... on: new ways of analysing data
@ast
Relationships between inhibiti ...... on: new ways of analysing data
@en
Relationships between inhibiti ...... on: new ways of analysing data
@nl
P2093
P2860
P1433
P1476
Relationships between inhibiti ...... on: new ways of analysing data
@en
P2093
A Cornish-Bowden
M L Cárdenas
P2860
P304
P356
10.1042/0264-6021:3570263
P407
P577
2001-07-01T00:00:00Z