Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenes
about
Identification of xenoestrogens in food additives by an integrated in silico and in vitro approachEstrogen receptor transcription and transactivation: Estrogen receptor alpha and estrogen receptor beta: regulation by selective estrogen receptor modulators and importance in breast cancer.The Concise Guide to PHARMACOLOGY 2013/14: nuclear hormone receptors.Genome-wide dynamics of chromatin binding of estrogen receptors alpha and beta: mutual restriction and competitive site selection.Virtual screening of the estrogen receptor.Estrogen receptor β ligands: recent advances and biomedical applications.Agonistic and antagonistic estrogens in licorice root (Glycyrrhiza glabra).Endocrine-responsive breast cancer and strategies for combating resistance.The 2010 Philip S. Portoghese Medicinal Chemistry Lectureship: addressing the "core issue" in the design of estrogen receptor ligandsIn vitro and in vivo molecular imaging of estrogen receptor α and β homo- and heterodimerization: exploration of new modes of receptor regulation.Divide and Conquer May Not Be the Optimal Approach to Retain the Desirable Estrogenic Attributes of the Cyclopia Nutraceutical Extract, SM6Met.Synthesis and biodistribution of fluorine-18-labeled fluorocyclofenils for imaging the estrogen receptorCoMSIA and docking study of rhenium based estrogen receptor ligand analogs.Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model.Synthesis and biological evaluation of two agents for imaging estrogen receptor β by positron emission tomography: challenges in PET imaging of a low abundance target.Metal complex SERMs (selective oestrogen receptor modulators). The influence of different metal units on breast cancer cell antiproliferative effects.Fluorine-substituted cyclofenil derivatives as estrogen receptor ligands: synthesis and structure-affinity relationship study of potential positron emission tomography agents for imaging estrogen receptors in breast cancer.Estrogen receptors alpha and beta in the rodent mammary gland.Importance of extranuclear estrogen receptor-alpha and membrane G protein-coupled estrogen receptor in pancreatic islet survivalCyclic Ketoximes as Estrogen Receptor β Selective Agonists.Disulfiram and its novel derivative sensitize prostate cancer cells to the growth regulatory mechanisms of the cell by re-expressing the epigenetically repressed tumor suppressor-estrogen receptor β.Estrogen receptor-alpha agonists promote angiogenesis in human myometrial microvascular endothelial cells.Metabolite ligands of estrogen receptor-beta reduce primate coronary hyperreactivity.Computational Insights into Ligand Selectivity of Estrogen Receptors from Pharmacophore Modeling.Multiple Routes to Oestrogen Antagonism.
P2860
Q24656051-643371B1-F972-4AB0-9320-CD057EBBDEABQ24800731-CA53DC5E-4B94-486A-AFBB-845D2B7A4E5FQ30486738-4A98765F-6CA4-414A-ADAD-CA46D78FB88BQ33576510-ECE26252-3604-4235-9B73-F7FC7AB4CCF1Q34619281-B75C0DF4-D7A2-4DE9-81D7-4B13FB354A7AQ35016384-209CF208-FBA1-4E7D-9A43-21C723C80DFBQ35072289-3320E627-B859-46A2-BB6A-D4385CEAC9E5Q35084786-46CE45C8-40B4-438A-B3FE-554DE6111E7BQ35148605-666AFB5D-F45E-4F57-9A88-EF452D740843Q35595730-41D2C7EC-9027-4982-9AFE-7082C88EE40DQ35712301-F02CF703-AEE1-4B02-824A-98D33E2F370CQ35940081-5171571E-9DDC-43DD-9F20-638215FD309EQ35971487-0DAB8776-4D67-48EB-8657-6C3CC799AB95Q36175547-A48E33C0-9A45-4B3F-827B-916F37A97445Q36301166-3ED0B970-1E9F-444B-BBBF-37C995389F2AQ36364465-023B67DB-B723-489A-9364-D5B873FECD7CQ36848788-B20E3C2E-A70D-4921-B863-42C0CF50C808Q37152373-49FF0A87-117D-4684-8CBF-91D4759055FEQ37360446-88A34338-A9F4-4E75-9809-EDA7EDA1E0E8Q38773922-08F324C2-9708-41B8-99E2-FDE347F58ACEQ38817309-234C4402-0B6D-4BF6-BCDA-44418FABEF35Q45176124-857E1CAA-FB8E-4F17-BACA-83E078F02FE5Q46731901-B9A38323-7ABE-41C4-A4DC-06FA85F5DB31Q54485705-2AC77B8C-C35E-4B0E-82B5-71B178060BB0Q55452150-061CEAE8-DC33-4C14-B2F3-20F93CFD2BAA
P2860
Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenes
description
1999 nî lūn-bûn
@nan
1999 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@ast
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@en
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@nl
type
label
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@ast
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@en
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@nl
prefLabel
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@ast
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@en
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@nl
P2093
P356
P1476
Estrogen receptor subtype-sele ...... 5,6,11, 12-tetrahydrochrysenes
@en
P2093
B S Katzenellenbogen
J A Katzenellenbogen
K E Carlson
P304
P356
10.1021/JM990101B
P407
P577
1999-07-01T00:00:00Z