Structure-activity relationships and binding mode of styrylquinolines as potent inhibitors of HIV-1 integrase and replication of HIV-1 in cell culture
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HIV-1 integrase catalytic core: molecular dynamics and simulated fluorescence decays.Inhibition of HIV-1 integrase by modified oligonucleotides derived from U5' LTR.HIV-1 IN inhibitors: 2010 update and perspectivesA cooperative and specific DNA-binding mode of HIV-1 integrase depends on the nature of the metallic cofactor and involves the zinc-containing N-terminal domain.Bicyclic hydroxy-1H-pyrrolopyridine-trione containing HIV-1 integrase inhibitors.Efficacy of orally administered 2-substituted quinolines in experimental murine cutaneous and visceral leishmaniases.Relationship between the oligomeric status of HIV-1 integrase on DNA and enzymatic activity.HIV-1 integrase and RNase H activities as therapeutic targets.Targeting HIV-1 integrase.Clinical Use of Inhibitors of HIV-1 Integration: Problems and Prospects.Authentic HIV-1 integrase inhibitors.Inhibitors of strand transfer that prevent integration and inhibit human T-cell leukemia virus type 1 early replication.Integrase and integration: biochemical activities of HIV-1 integrase.HIV-1 integrase inhibitors: a review of their chemical development.Drug design using comparative molecular surface analysis.Comparison of Newly Assembled Full Length HIV-1 Integrase With Prototype Foamy Virus Integrase: Structure-Function Prospective.Bioactivity-guided isolation of anticancer agents from Bauhinia kockiana Korth.Different Pathways Leading to Integrase Inhibitors ResistanceSupport Vector Machine (SVM) Models for Predicting Inhibitors of the 3' Processing Step of HIV-1 Integrase.Styrylquinolines, integrase inhibitors acting prior to integration: a new mechanism of action for anti-integrase agents.In vitro activities of new 2-substituted quinolines against Leishmania donovani.Computational models on quantitative prediction of bioactivity of HIV-1 integrase 3' processing inhibitors.3-[(E)-2-(5,7-Dichloro-8-hydroxy-quinolin-2-yl)vin-yl]-4-hydroxy-phenyl acetate.Dual Behavior of Iodine Species in Condensation of Anilines and Vinyl Ethers Affording 2-Methylquinolines.A general three-step one-pot synthesis of novel (E)-6-chloro-2-(aryl/hetarylvinyl)quinoline-3-carboxylic acids.3D-QSAR studies of quinoline ring derivatives as HIV-1 integrase inhibitors.
P2860
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P2860
Structure-activity relationships and binding mode of styrylquinolines as potent inhibitors of HIV-1 integrase and replication of HIV-1 in cell culture
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2000 nî lūn-bûn
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2000 թուականի Ապրիլին հրատարակուած գիտական յօդուած
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2000 թվականի ապրիլին հրատարակված գիտական հոդված
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2000年の論文
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2000年学术文章
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2000年学术文章
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2000年学术文章
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Structure-activity relationshi ...... ation of HIV-1 in cell culture
@ast
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@en
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@nl
type
label
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@ast
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@en
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@nl
prefLabel
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@ast
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@en
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@nl
P2093
P356
P1476
Structure-activity relationshi ...... ation of HIV-1 in cell culture
@en
P2093
D Desmaële
J F Mouscadet
J d'Angelo
P304
P356
10.1021/JM990467O
P407
P577
2000-04-20T00:00:00Z