Human A(2A) adenosine receptors: high-affinity agonist binding to receptor-G protein complexes containing Gbeta(4).
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Agonist-bound adenosine A2A receptor structures reveal common features of GPCR activationThe A3 adenosine receptor agonist CP-532,903 [N6-(2,5-dichlorobenzyl)-3'-aminoadenosine-5'-N-methylcarboxamide] protects against myocardial ischemia/reperfusion injury via the sarcolemmal ATP-sensitive potassium channelA2A receptors in inflammation and injury: lessons learned from transgenic animalsStructural determinants involved in the formation and activation of G protein betagamma dimers.Attenuation of gastric mucosal inflammation induced by aspirin through activation of A2A adenosine receptor in rats.The infarct-sparing effect of IB-MECA against myocardial ischemia/reperfusion injury in mice is mediated by sequential activation of adenosine A3 and A 2A receptors.Activation of A2A adenosine receptors inhibits expression of alpha 4/beta 1 integrin (very late antigen-4) on stimulated human neutrophils.Adenosine A2A receptor activation reduces recurrence and mortality from Clostridium difficile infection in mice following vancomycin treatment.Binding of β4γ5 by adenosine A1 and A2A receptors determined by stable isotope labeling with amino acids in cell culture and mass spectrometry.Adenosine A2A receptor signaling and golf assembly show a specific requirement for the gamma7 subtype in the striatumLipopolysaccharide rapidly modifies adenosine receptor transcripts in murine and human macrophages: role of NF-kappaB in A(2A) adenosine receptor induction.Adenosine A2A receptor activation reduces infarct size in the isolated, perfused mouse heart by inhibiting resident cardiac mast cell degranulation.The allosteric enhancer PD81,723 increases chimaeric A1/A2A adenosine receptor coupling with GsCharacterization of the A2B adenosine receptor from mouse, rabbit, and dog.Nanobodies to Study G Protein-Coupled Receptor Structure and Function.Programmable nanoscaffolds that control ligand display to a G-protein-coupled receptor in membranes to allow dissection of multivalent effects.Thermostabilisation of an agonist-bound conformation of the human adenosine A(2A) receptor.Functional coupling of the Galpha(olf) variant XLGalpha(olf) with the human adenosine A2A receptor.A role for the low-affinity A2B adenosine receptor in regulating superoxide generation by murine neutrophilsAdenosine receptor agonists: from basic medicinal chemistry to clinical development.Protection from myocardial ischemia/reperfusion injury by a positive allosteric modulator of the A₃ adenosine receptor.Mechanisms of modulation of cytokine release by human cord blood monocytes exposed to high concentrations of caffeineNovel approaches for targeting the adenosine A2A receptor.Inhibition of sequestration of human B2 bradykinin receptor by phenylarsine oxide or sucrose allows determination of a receptor affinity shift and ligand dissociation in intact cells.Structure of the adenosine A(2A) receptor bound to an engineered G protein.Characterization of human and rodent native and recombinant adenosine A(2B) receptors by radioligand binding studies.Regulation of adenosine receptor subtypes during cultivation of human monocytes: role of receptors in preventing lipopolysaccharide-triggered respiratory burst.Selectivity is species-dependent: Characterization of standard agonists and antagonists at human, rat, and mouse adenosine receptors.Role of extracellular cysteine residues in the adenosine A2A receptor.A3 adenosine receptor agonist IB-MECA reduces myocardial ischemia-reperfusion injury in dogsSelective adenosine A receptor agonist, ATL-146e, attenuates stress-induced gastric lesions in rats.Species differences and mechanism of action of A3 adenosine receptor allosteric modulators.Human Adenosine A2A Receptor: Molecular Mechanism of Ligand Binding and Activation.
P2860
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P2860
Human A(2A) adenosine receptors: high-affinity agonist binding to receptor-G protein complexes containing Gbeta(4).
description
2002 nî lūn-bûn
@nan
2002 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2002 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2002年の論文
@ja
2002年論文
@yue
2002年論文
@zh-hant
2002年論文
@zh-hk
2002年論文
@zh-mo
2002年論文
@zh-tw
2002年论文
@wuu
name
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@ast
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@en
type
label
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@ast
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@en
prefLabel
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@ast
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@en
P2093
P356
P1476
Human A(2A) adenosine receptor ...... complexes containing Gbeta(4).
@en
P2093
Jayson M Rieger
Joel Linden
Lauren J Murphree
Melissa A Marshall
Timothy L MacDonald
P304
P356
10.1124/MOL.61.2.455
P577
2002-02-01T00:00:00Z