Structure-activity relationships for a series of quinoline-based compounds active against replicating and nonreplicating Mycobacterium tuberculosis.
about
Structure-activity relationship of new anti-tuberculosis agents derived from oxazoline and oxazole benzyl esters.A novel quinoline derivative that inhibits mycobacterial FtsZ.Synthesis and SAR studies of novel 6,7,8-substituted 4-substituted benzyloxyquinolin-2(1H)-one derivatives for anticancer activityPutting Tuberculosis (TB) To Rest: Transformation of the Sleep Aid, Ambien, and "Anagrams" Generated Potent Antituberculosis Agents.Library of diversely substituted 2-(quinolin-4-yl)imidazolines delivers novel non-cytotoxic antitubercular leads.Pyrido[1,2-a]benzimidazole-based agents active against tuberculosis (TB), multidrug-resistant (MDR) TB and extensively drug-resistant (XDR) TB2-(Quinolin-4-yloxy)acetamides Are Active against Drug-Susceptible and Drug-Resistant Mycobacterium tuberculosis Strains.Chemotherapeutic interventions against tuberculosisStructural Simplification of Bedaquiline: the Discovery of 3-(4-(N,N-Dimethylaminomethyl)phenyl)quinoline-Derived Antitubercular Lead Compounds.Recent advances in the design and synthesis of heterocycles as anti-tubercular agents.Antituberculosis drug research: a critical overview.New substituted benzimidazole derivatives: a patent review (2010 - 2012).N-(Prop-2-yn-1-yl)-1,3-benzothia-zol-2-amineNitazoxanide Disrupts Membrane Potential and Intrabacterial pH Homeostasis of Mycobacterium tuberculosis.Targeting Phenotypically Tolerant Mycobacterium tuberculosis.1-Prop-2-ynyl-1H-benzimidazol-2-amineOne-pot tandem Ugi-4CR/S(N)Ar approach to highly functionalized quino[2,3-b][1,5]benzoxazepines.Methyl 2-{[2,8-bis-(trifluoro-meth-yl)quinolin-4-yl]-oxy}acetate.Quinoline: A versatile heterocyclictert-Butyl N-{2-[bis-(prop-2-yn-1-yl)amino]-phen-yl}carbamate.Cu-catalyzed tandem reactions of fluorinated alkynes with sulfonyl azides en route to 2-trifluoromethylquinolines.A Dy4 single-molecule magnet and its Gd(iii), Tb(iii), Ho(iii), and Er(iii) analogues encapsulated by an 8-hydroxyquinoline Schiff base derivative and β-diketonate coligand.Iodine mediated oxidative cross-coupling of unprotected anilines and heteroarylation of benzothiazoles with 2-methylquinoline.Palladium-catalyzed intermolecular oxidative cyclization of N-aryl enamines with isocyanides through double sp(2) C-H bonds cleavage: facile synthesis of 4-aminoquinoline derivatives.Visible-light-induced radical cyclization of trifluoroacetimidoyl chlorides with alkynes: catalytic synthesis of 2-trifluoromethyl quinolines.Synthesis, antimicrobial, and antiviral activities of some new 5-sulphonamido-8-hydroxyquinoline derivatives.Activity of mefloquine and mefloquine derivatives against Echinococcus multilocularisCopper-catalyzed synthesis of quinoline derivatives via tandem Knoevenagel condensation, amination and cyclizationBasic hydrolysis of quinolinyl N,N-dimethylcarbamates: a two-step mechanism
P2860
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P2860
Structure-activity relationships for a series of quinoline-based compounds active against replicating and nonreplicating Mycobacterium tuberculosis.
description
2009 nî lūn-bûn
@nan
2009 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@ast
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@en
type
label
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@ast
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@en
prefLabel
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@ast
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@en
P2093
P356
P1476
Structure-activity relationshi ...... ng Mycobacterium tuberculosis.
@en
P2093
Alan P Kozikowski
Annamaria Lilienkampf
Baojie Wan
Jialin Mao
Yuehong Wang
P304
P356
10.1021/JM900003C
P407
P577
2009-04-01T00:00:00Z