Design, Synthesis, and Biological Evaluation of PKD Inhibitors.

Design, Synthesis, and Biological Evaluation of PKD Inhibitors.

Item
http://www.wikidata.org/entity/Q30428751
Protein kinase D enzymes: novel kinase targets in pancreatic cancerA targeted library screen reveals a new inhibitor scaffold for protein kinase DProtein Kinase Inhibitors CK59 and CID755673 Alter Primary Human NK Cell Effector FunctionsSustained protein kinase D activation mediates respiratory syncytial virus-induced airway barrier disruption.In vitro cytotoxicity, pharmacokinetics, tissue distribution, and metabolism of small-molecule protein kinase D inhibitors, kb-NB142-70 and kb-NB165-09, in mice bearing human cancer xenografts.A bifunctional dimethylsulfoxide substitute enhances the aqueous solubility of small organic molecules.New pyrazolopyrimidine inhibitors of protein kinase d as potent anticancer agents for prostate cancer cellsPromiscuous actions of small molecule inhibitors of the protein kinase D-class IIa HDAC axis in striated muscleFunctional and therapeutic significance of protein kinase D enzymes in invasive breast cancer.Regulation of membrane KCNQ1/KCNE1 channel density by sphingomyelin synthase 1.Protein kinase D isoforms: new targets for therapy in invasive breast cancers?Protein kinase D signaling in cancer: A friend or foe?An uncharged oxetanyl sulfoxide as a covalent modifier for improving aqueous solubility.Protein kinase D2: a versatile player in cancer biology.Enantioselective Phosphine-Catalyzed Formal [4+4] Annulation of α,β-Unsaturated Imines and Allene Ketones: Construction of Eight-Membered Rings.Diversity-oriented synthesis of fused thioglycosyl benzo[e][1,4]oxathiepin-5-ones and benzo[f][1,4]thiazepin-5(2H)-ones by a sequence of palladium-catalyzed glycosyl thiol arylation and deprotection-lactonization reactions.Hippocampal protein kinase D1 is necessary for DHPG-induced learning and memory impairments in rats.
P2860

Design, Synthesis, and Biological Evaluation of PKD Inhibitors.

Item
http://www.wikidata.org/entity/Q30428751
description
2011 nî lūn-bûn
@nan
2011 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@ast
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@en
type
label
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@ast
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@en
prefLabel
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@ast
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@en
P1433
P1476
P2093
P2860
P304
P31
P356
P433
P478
P50
P577
P5875
P698
P932
P356
P1433
P1476
Design, Synthesis, and Biological Evaluation of PKD Inhibitors.
@en
P2093
P2860
P304
P31
P356
10.3390/PHARMACEUTICS3020186
P433
P478
P50
P577
P5875
P698
P932