Kinome-wide activity modeling from diverse public high-quality data sets
about
Comparability of mixed IC₅₀ data - a statistical analysisHigh quality, small molecule-activity datasets for kinase researchUNC2025, a potent and orally bioavailable MER/FLT3 dual inhibitor.Large-scale integration of small molecule-induced genome-wide transcriptional responses, Kinome-wide binding affinities and cell-growth inhibition profiles reveal global trends characterizing systems-level drug action.Chemical interrogation of the neuronal kinome using a primary cell-based screening assay.Screening of cell cycle fusion proteins to identify kinase signaling networksLarge-Scale Computational Screening Identifies First in Class Multitarget Inhibitor of EGFR Kinase and BRD4.Rational Polypharmacology: Systematically Identifying and Engaging Multiple Drug Targets To Promote Axon Growth.Computational methods for analysis and inference of kinase/inhibitor relationships.Epigenetic pathways and glioblastoma treatment: insights from signaling cascades.Unprecedently Large-Scale Kinase Inhibitor Set Enabling the Accurate Prediction of Compound-Kinase Activities: A Way toward Selective Promiscuity by Design?SimBoost: a read-across approach for predicting drug-target binding affinities using gradient boosting machines.Drug Repositioning in Glioblastoma: A Pathway Perspective.
P2860
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P2860
Kinome-wide activity modeling from diverse public high-quality data sets
description
2013 nî lūn-bûn
@nan
2013 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
Kinome-wide activity modeling from diverse public high-quality data sets
@ast
Kinome-wide activity modeling from diverse public high-quality data sets
@en
type
label
Kinome-wide activity modeling from diverse public high-quality data sets
@ast
Kinome-wide activity modeling from diverse public high-quality data sets
@en
prefLabel
Kinome-wide activity modeling from diverse public high-quality data sets
@ast
Kinome-wide activity modeling from diverse public high-quality data sets
@en
P2860
P356
P1476
Kinome-wide activity modeling from diverse public high-quality data sets
@en
P2093
Stephan C Schürer
Steven M Muskal
P2860
P356
10.1021/CI300403K
P577
2013-01-09T00:00:00Z