Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography.
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Adenosine A2A receptors and basal ganglia physiologyRecent developments in adenosine receptor ligands and their potential as novel drugsAdenosine 2A receptor availability in dyskinetic and nondyskinetic patients with Parkinson diseaseThe Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsQuinolinic acid induced neurodegeneration in the striatum: a combined in vivo and in vitro analysis of receptor changes and microglia activation.Synthesis and evaluation of 1,2,4-triazolo[1,5-c]pyrimidine derivatives as A2A receptor-selective antagonistsMolecular probes for the A2A adenosine receptor based on a pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine scaffoldIsothermal chemical denaturation to determine binding affinity of small molecules to G-protein coupled receptors.Hide and seek: a comparative autoradiographic in vitro investigation of the adenosine A3 receptorPyrazolo derivatives as potent adenosine receptor antagonists: an overview on the structure-activity relationshipsBiosensor-based affinities and binding kinetics of small molecule antagonists to the adenosine A(2A) receptor reconstituted in HDL like particles.Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: A complete structure-activity profile.Application of the functionalized congener approach to dendrimer-based signaling agents acting through A(2A) adenosine receptors.History and perspectives of A2A adenosine receptor antagonists as potential therapeutic agents.Potential Therapeutic Applications of Adenosine A2A Receptor Ligands and Opportunities for A2A Receptor Imaging.An old friend with new skills: Imiquimod as novel inhibitor of Hedgehog signaling in basal cell carcinoma.The adenosine A2A receptor antagonist ZM241385 enhances neuronal survival after oxygen-glucose deprivation in rat CA1 hippocampal slices.In vivo labelling of the adenosine A2A receptor in mouse brain using the selective antagonist [3H]SCH 58261.Evaluation of [4-O-methyl-(11)C]KW-6002 as a potential PET ligand for mapping central adenosine A(2A) receptors in rats.In Vivo PET Imaging of Adenosine 2A Receptors in Neuroinflammatory and Neurodegenerative Disease.Photoaffinity Labeling of the Human A2A Adenosine Receptor and Cross-link Position Analysis by Mass Spectrometry.The prediction of blood-tissue partitions, water-skin partitions and skin permeation for agrochemicals.PBF509, an Adenosine A Receptor Antagonist With Efficacy in Rodent Models of Movement Disorders
P2860
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P2860
Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography.
description
2000 nî lūn-bûn
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2000 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի նոյեմբերին հրատարակված գիտական հոդված
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2000年の論文
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2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
Design, radiosynthesis, and bi ...... positron emission tomography.
@ast
Design, radiosynthesis, and bi ...... positron emission tomography.
@en
type
label
Design, radiosynthesis, and bi ...... positron emission tomography.
@ast
Design, radiosynthesis, and bi ...... positron emission tomography.
@en
prefLabel
Design, radiosynthesis, and bi ...... positron emission tomography.
@ast
Design, radiosynthesis, and bi ...... positron emission tomography.
@en
P2093
P356
P1476
Design, radiosynthesis, and bi ...... positron emission tomography.
@en
P2093
Baraldi PG
Cacciari B
Carpinelli A
Matarrese M
Monopoli A
Moresco RM
Simonelli P
P304
P356
10.1021/JM0009843
P407
P577
2000-11-01T00:00:00Z