"Carba"-analogues of fentanyl are opioid receptor agonists.
about
'Carba'-carfentanil (trans isomer): a μ opioid receptor (MOR) partial agonist with a distinct binding mode.Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications.Discovery of 5-substituted tetrahydronaphthalen-2yl-methyl with N-phenyl-N-(piperidin-4-yl)propionamide derivatives as potent opioid receptor ligands.Design synthesis and structure-activity relationship of 5-substituted (tetrahydronaphthalen-2yl)methyl with N-phenyl-N-(piperidin-2-yl)propionamide derivatives as opioid ligandsTryptophan-Containing Non-Cationizable Opioid Peptides - a new chemotype with unusual structure and in vivo activity.A systematic analysis of atomic protein-ligand interactions in the PDB.The inverse type II β-turn on D-Trp-Phe, a pharmacophoric motif for MOR agonists.
P2860
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P2860
"Carba"-analogues of fentanyl are opioid receptor agonists.
description
2010 nî lūn-bûn
@nan
2010 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
"Carba"-analogues of fentanyl are opioid receptor agonists.
@ast
"Carba"-analogues of fentanyl are opioid receptor agonists.
@en
type
label
"Carba"-analogues of fentanyl are opioid receptor agonists.
@ast
"Carba"-analogues of fentanyl are opioid receptor agonists.
@en
prefLabel
"Carba"-analogues of fentanyl are opioid receptor agonists.
@ast
"Carba"-analogues of fentanyl are opioid receptor agonists.
@en
P2093
P2860
P356
P1476
"Carba"-analogues of fentanyl are opioid receptor agonists.
@en
P2093
Brian C Wilkes
Carole Lemieux
Grazyna Weltrowska
Jianxin Guo
Nga N Chung
Peter W Schiller
P2860
P304
P356
10.1021/JM9019068
P407
P577
2010-04-01T00:00:00Z