Probes for the cocaine receptor. Potentially irreversible ligands for the dopamine transporter.

Probes for the cocaine receptor. Potentially irreversible ligands for the dopamine transporter.

Item
http://www.wikidata.org/entity/Q33987010
Tropane and Granatane Alkaloid Biosynthesis: A Systematic AnalysisDevelopment of 3-phenyltropane analogues with high affinity for the dopamine and serotonin transporters and low affinity for the norepinephrine transporter.Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling.Evolution of a Compact Photoprobe for the Dopamine Transporter Based on (±)-threo-Methylphenidate.Computational and biochemical docking of the irreversible cocaine analog RTI 82 directly demonstrates ligand positioning in the dopamine transporter central substrate-binding site.Synthesis and structure-activity relationship of 3beta-(4-alkylthio, -methylsulfinyl, and -methylsulfonylphenyl)tropane and 3beta-(4-alkylthiophenyl)nortropane derivatives for monoamine transporters.The last step in cocaine biosynthesis is catalyzed by a BAHD acyltransferase.Novel Azido-Iodo Photoaffinity Ligands for the Human Serotonin Transporter Based on the Selective Serotonin Reuptake Inhibitor (S)-Citalopram.Irreversible binding of a novel phenylisothiocyanate tropane analog to monoamine transporters in rat brainAnti-drug vaccines to treat substance abuse.A novel photoaffinity ligand for the dopamine transporter based on pyrovalerone.Effects of ginseng saponin on acute cocaine-induced alterations in evoked dopamine release and uptake in rat brain nucleus accumbens.Recovery of dopamine neuronal transporter but lack of change of its mRNA in substantia nigra after inactivation by a new irreversible inhibitor characterized in vitro and ex vivo in the rat.Differential time-course profiles of dopamine release and uptake changes induced by three dopamine uptake inhibitors.Phorbol ester induced trafficking-independent regulation and enhanced phosphorylation of the dopamine transporter associated with membrane rafts and cholesterol.Localization of cocaine analog [125I]RTI 82 irreversible binding to transmembrane domain 6 of the dopamine transporter.RTI-352: a 3 alpha analogue of RTI-55 as an in vivo dopamine transporter binding ligand.
P2860

Probes for the cocaine receptor. Potentially irreversible ligands for the dopamine transporter.

Item
http://www.wikidata.org/entity/Q33987010
description
1992 nî lūn-bûn
@nan
1992 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
1992 թվականի մայիսին հրատարակված գիտական հոդված
@hy
1992年の論文
@ja
1992年論文
@yue
1992年論文
@zh-hant
1992年論文
@zh-hk
1992年論文
@zh-mo
1992年論文
@zh-tw
1992年论文
@wuu
name
Probes for the cocaine recepto ...... for the dopamine transporter.
@ast
Probes for the cocaine recepto ...... for the dopamine transporter.
@en
type
label
Probes for the cocaine recepto ...... for the dopamine transporter.
@ast
Probes for the cocaine recepto ...... for the dopamine transporter.
@en
prefLabel
Probes for the cocaine recepto ...... for the dopamine transporter.
@ast
Probes for the cocaine recepto ...... for the dopamine transporter.
@en
P1433
P1476
P2093
P304
P31
P356
P407
P433
P478
P577
P698
P356
P1433
P1476
Probes for the cocaine recepto ...... for the dopamine transporter.
@en
P2093
P304
P31
P356
P407
P433
P478
P577
P698