Pharmacology of putative selective hBRS-3 receptor agonists for human bombesin receptors (BnR): affinities, potencies and selectivity in multiple native and BnR transfected cells.
about
Insights into bombesin receptors and ligands: Highlighting recent advancesBombesin receptor subtype 3 as a potential target for obesity and diabetes.Novel chiral-diazepines function as specific, selective receptor agonists with variable coupling and species variability in human, mouse and rat BRS-3 receptor cells.Bombesin receptor subtype-3 agonists stimulate the growth of lung cancer cells and increase EGF receptor tyrosine phosphorylation.The molecular basis for high affinity of a universal ligand for human bombesin receptor (BnR) family members.Comparative pharmacology of bombesin receptor subtype-3, nonpeptide agonist MK-5046, a universal peptide agonist, and peptide antagonist Bantag-1 for human bombesin receptorsBombesin related peptides/receptors and their promising therapeutic roles in cancer imaging, targeting and treatment.Gastrin-releasing peptide receptor mediates the excitation of preoptic GABAergic neurons by bombesin.A selective human bombesin receptor subtype-3 peptide agonist mediates CREB phosphorylation and transactivation.Molecular basis for high affinity and selectivity of peptide antagonist, Bantag-1, for the orphan BB3 receptor.A possible new target in lung-cancer cells: The orphan receptor, bombesin receptor subtype-3.
P2860
Q28081153-C2B64B82-9C0E-42D6-8C3B-17EE7CA08909Q33637115-7B27566A-56D9-4B5D-B4DE-3795E1469768Q33771938-1AA114FA-D30C-4C6C-AD04-CA623CBD671DQ35154082-B71C870E-8503-41B9-AB4E-52AF19CBB56AQ36208460-CC09D24E-3376-4121-9FE6-DF22C57BE71BQ37193224-3495E790-15B4-4334-8950-F79404380C42Q38776596-9CF292E8-C53F-4F76-B959-44D72CEF3867Q39331675-E8AB6AF1-2D71-490E-B46C-A40EB7091B01Q39435556-9A7AF6A2-4B31-49B6-83A9-F55C53FFB010Q42365925-12E0D100-D148-4A79-98FF-51A8A6121BE2Q50149052-756CB0CC-1A35-431F-B11A-BFCD465DBA18
P2860
Pharmacology of putative selective hBRS-3 receptor agonists for human bombesin receptors (BnR): affinities, potencies and selectivity in multiple native and BnR transfected cells.
description
2010 nî lūn-bûn
@nan
2010 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Pharmacology of putative selec ...... ive and BnR transfected cells.
@ast
Pharmacology of putative selec ...... ive and BnR transfected cells.
@en
Pharmacology of putative selec ...... ive and BnR transfected cells.
@nl
type
label
Pharmacology of putative selec ...... ive and BnR transfected cells.
@ast
Pharmacology of putative selec ...... ive and BnR transfected cells.
@en
Pharmacology of putative selec ...... ive and BnR transfected cells.
@nl
prefLabel
Pharmacology of putative selec ...... ive and BnR transfected cells.
@ast
Pharmacology of putative selec ...... ive and BnR transfected cells.
@en
Pharmacology of putative selec ...... ive and BnR transfected cells.
@nl
P2093
P2860
P1433
P1476
Pharmacology of putative selec ...... ive and BnR transfected cells.
@en
P2093
Alessia Di Florio
David H Coy
Hirotsugu Uehara
Robert T Jensen
Samuel A Mantey
Terry W Moody
Veronica Sancho
P2860
P304
P356
10.1016/J.PEPTIDES.2010.04.023
P577
2010-05-12T00:00:00Z