Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
about
Hotspot mutations in KIT receptor differentially modulate its allosterically coupled conformational dynamics: impact on activation and drug sensitivityEfficacy and safety of motesanib, an oral inhibitor of VEGF, PDGF, and Kit receptors, in patients with imatinib-resistant gastrointestinal stromal tumors.Limited Tumor Tissue Drug Penetration Contributes to Primary Resistance against Angiogenesis InhibitorsMolecular mechanisms of drug resistance in tyrosine kinases cAbl and cKit.Systemic therapy for advanced gastrointestinal stromal tumors: beyond imatinib.Treatments for gastrointestinal stromal tumors that are resistant to standard therapies.
P2860
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
description
2010 nî lūn-bûn
@nan
2010 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@ast
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@en
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@nl
type
label
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@ast
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@en
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@nl
prefLabel
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@ast
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@en
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@nl
P2093
P2860
P356
P1476
Motesanib inhibits Kit mutations associated with gastrointestinal stromal tumors.
@en
P2093
Andrew S Tasker
Angelo Baher
Anthony Polverino
Lisa Renshaw-Gegg
Paul E Hughes
Raffi Manoukian
Sean Caenepeel
Tammy L Bush
Will Baron
P2860
P2888
P356
10.1186/1756-9966-29-96
P577
2010-07-15T00:00:00Z
P5875
P6179
1020911816