Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
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Histamine and Skin Barrier: Are Histamine Antagonists Useful for the Prevention or Treatment of Atopic Dermatitis?International Union of Basic and Clinical Pharmacology. XCVIII. Histamine ReceptorsLuciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readoutsThe Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsImplementation of a fluorescence-based screening assay identifies histamine H3 receptor antagonists clobenpropit and iodophenpropit as subunit-selective N-methyl-D-aspartate receptor antagonists.Histamine H4-receptors inhibit mast cell renin release in ischemia/reperfusion via protein kinase C ε-dependent aldehyde dehydrogenase type-2 activationHistamine receptors and cancer pharmacology.H3 receptors and pain modulation: peripheral, spinal, and brain interactions.Brain P450 epoxygenase activity is required for the antinociceptive effects of improgan, a nonopioid analgesic.The role of histamine H4 receptor in immune and inflammatory disordersIdentification of histamine receptors and effects of histamine on murine and simian colonic excitability.Histamine 3 receptor activation reduces the expression of neuronal angiotensin II type 1 receptors in the heart.Histamine induces proliferation in keratinocytes from patients with atopic dermatitis through the histamine 4 receptor.CC12, a high-affinity ligand for [3H]cimetidine binding, is an improgan antagonist.Potentiation of NF-kappaB-dependent transcription and inflammatory mediator release by histamine in human airway epithelial cellsAntinociceptive activity of furan-containing congeners of improgan and ranitidine.Synthesis of Substituted 2-phenylhistamines via a Microwave Promoted Suzuki Coupling.Natriuretic peptide-induced catecholamine release from cardiac sympathetic neurons: inhibition by histamine H3 and H4 receptor activation.Histamine H4 receptor antagonists as potent modulators of mammalian vestibular primary neuron excitability.The histamine H4 receptor in autoimmune disease.Effects of histamine on cultured interstitial cells of cajal in murine small intestine.Small mouse cholangiocytes proliferate in response to H1 histamine receptor stimulation by activation of the IP3/CaMK I/CREB pathway.Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas.Therapeutic potential of histamine H₄ receptor agonists in triple-negative human breast cancer experimental model.Molecular and cellular analysis of human histamine receptor subtypes.Molecular and biochemical pharmacology of the histamine H4 receptor.Histamine H4 receptor ligands and their potential therapeutic applications.Histamine H3 and H4 receptors as novel drug targets.Environmental stressors and neurobiological features of marine teleosts: histamine receptors as targets.Histamine H4 receptor ligands and their potential therapeutic applications: an update.(11) C-labeled and (18) F-labeled PET ligands for subtype-specific imaging of histamine receptors in the brain.Histamine H4 receptor ligands: future applications and state of art.The histamine H4 receptor: from orphan to the clinic.Activation of the ileal neuroendocrine tumor cell line P-STS by acetylcholine is amplified by histamine: role of H3R and H4R.The Histamine H3 Receptor: Structure, Pharmacology, and Function.Clinical Development of Histamine H4 Receptor Antagonists.Pharmacological Characterization of Human Histamine Receptors and Histamine Receptor Mutants in the Sf9 Cell Expression System.Histamine induces chemotaxis and phagocytosis in murine bone marrow-derived macrophages and RAW 264.7 macrophage-like cells via histamine H4-receptor.Profiling of histamine H4 receptor agonists in native human monocytes.Molecular mechanism of histamine clearance by primary human astrocytes.
P2860
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P2860
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
description
2005 nî lūn-bûn
@nan
2005 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2005年の論文
@ja
2005年論文
@yue
2005年論文
@zh-hant
2005年論文
@zh-hk
2005年論文
@zh-mo
2005年論文
@zh-tw
2005年论文
@wuu
name
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@ast
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@en
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@nl
type
label
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@ast
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@en
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@nl
prefLabel
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@ast
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@en
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@nl
P2093
P356
P1476
Evaluation of histamine H1-, H ...... selective H4 receptor agonist.
@en
P2093
Herman D Lim
Remko A Bakker
Richard M van Rijn
P304
P356
10.1124/JPET.105.087965
P407
P577
2005-06-09T00:00:00Z