Pharmacological properties of GABAA receptors containing gamma1 subunits.
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International Union of Pharmacology. LXX. Subtypes of gamma-aminobutyric acid(A) receptors: classification on the basis of subunit composition, pharmacology, and function. UpdateAssociations among GABRG1, level of response to alcohol, and drinking behaviorsMarkers in the 5'-region of GABRG1 associate to alcohol dependence and are in linkage disequilibrium with markers in the adjacent GABRA2 geneEfficient modulation of γ-aminobutyric acid type A receptors by piperine derivatives.HPLC-based activity profiling: discovery of piperine as a positive GABA(A) receptor modulator targeting a benzodiazepine-independent binding site.Esters of valerenic acid as potential prodrugs.The Genetics, Neurogenetics and Pharmacogenetics of AddictionMolecular tools for GABAA receptors: High affinity ligands for β1-containing subtypes.Valerenic acid derivatives as novel subunit-selective GABAA receptor ligands - in vitro and in vivo characterization.Tolerance to the rate-increasing and not rate-decreasing effects of pregnanolone in ratsGenetic association of recovery from eating disorders: the role of GABA receptor SNPs.Automated fast perfusion of Xenopus oocytes for drug screeningInsights into structure-activity relationship of GABAA receptor modulating coumarins and furanocoumarins.HPLC-based activity profiling approach for the discovery of GABAA receptor ligands using an automated two microelectrode voltage clamp assay on Xenopus oocytes.HPLC-based activity profiling for GABAA receptor modulators from the traditional Chinese herbal drug Kushen (Sophora flavescens root).Positive GABA(A) receptor modulators from Acorus calamus and structural analysis of (+)-dioxosarcoguaiacol by 1D and 2D NMR and molecular modelingIdentification of GABA A receptor modulators in Kadsura longipedunculata and assignment of absolute configurations by quantum-chemical ECD calculationsFunctional characterization of the 1,5-benzodiazepine clobazam and its major active metabolite N-desmethylclobazam at human GABA(A) receptors expressed in Xenopus laevis oocytes.Analysis of β-Subunit-dependent GABAA Receptor Modulation and Behavioral Effects of Valerenic Acid Derivatives.Loss of functional GABA(A) receptors in the Alzheimer diseased brain.Comparison of cell expression formats for the characterization of GABA(A) channels using a microfluidic patch clamp system.Estimating the efficiency of benzodiazepines on GABA(A) receptors comprising gamma1 or gamma2 subunits.Zolpidem is a potent stoichiometry-selective modulator of α1β3 GABAA receptors: evidence of a novel benzodiazepine site in the α1-α1 interface.GABAA receptor modulation by piperine and a non-TRPV1 activating derivativeIdentification of the putative binding pocket of valerenic acid on GABAA receptors using docking studies and site-directed mutagenesis.Function and modulation of delta-containing GABA(A) receptorsFast and Slow Inhibition in the Visual Thalamus Is Influenced by Allocating GABAA Receptors with Different γ Subunits.A novel GABA(A) receptor pharmacology: drugs interacting with the α(+) β(-) interface.The behavioral pharmacology of zolpidem: evidence for the functional significance of α1-containing GABA(A) receptors.Clobazam as an adjunctive therapy in treating seizures associated with Lennox-Gastaut syndrome.Optimizing the expression of recombinant alphabetagamma GABAA receptors in HEK293 cells for high-throughput screening.GABAA receptors containing gamma1 subunits contribute to inhibitory transmission in the central amygdala.Benzodiazepine-site pharmacology on GABAA receptors in histaminergic neuronsα2 Subunit-Containing GABAA Receptor Subtypes Are Upregulated and Contribute to Alcohol-Induced Functional Plasticity in the Rat Hippocampus.GABA Receptors and the Pharmacology of Sleep.Analysis of γ-aminobutyric acid (GABA) type A receptor subtypes using isosteric and allosteric ligands.PharmGKB summary: clobazam pathway, pharmacokinetics.Sigmoid colon mucosal gene expression supports alterations of neuronal signaling in irritable bowel syndrome with constipation.
P2860
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P2860
Pharmacological properties of GABAA receptors containing gamma1 subunits.
description
2005 nî lūn-bûn
@nan
2005 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2005年の論文
@ja
2005年論文
@yue
2005年論文
@zh-hant
2005年論文
@zh-hk
2005年論文
@zh-mo
2005年論文
@zh-tw
2005年论文
@wuu
name
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@ast
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@en
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@nl
type
label
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@ast
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@en
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@nl
prefLabel
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@ast
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@en
Pharmacological properties of GABAA receptors containing gamma1 subunits.
@nl
P2093
P356
P1476
Pharmacological properties of GABAA receptors containing gamma1 subunits
@en
P2093
P304
P356
10.1124/MOL.105.017236
P577
2005-11-04T00:00:00Z