Probes for narcotic receptor mediated phenomena. 41. Unusual inverse μ-agonists and potent μ-opioid antagonists by modification of the N-substituent in enantiomeric 5-(3-hydroxyphenyl)morphans

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description

2011 nî lūn-bûn

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2011 թուականի Յունուարին հրատարակուած գիտական յօդուած

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2011 թվականի հունվարին հրատարակված գիտական հոդված

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2011年の論文

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2011年論文

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2011年論文

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2011年論文

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2011年論文

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2011年論文

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2011年论文

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Probes for narcotic receptor m ...... substituent in enantiomeric 5-

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Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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type

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Probes for narcotic receptor m ...... substituent in enantiomeric 5-

@nl

Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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Probes for narcotic receptor m ...... substituent in enantiomeric 5-

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Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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P1476

Probes for narcotic receptor m ...... ic 5-(3-hydroxyphenyl)morphans

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P2093

Arthur E Jacobson

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Christina M Dersch

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Kejun Cheng

http://www.w3.org/2001/XMLSchema#string

Kenner C Rice

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Richard B Rothman

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Yong Sok Lee

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P2860

Opioid peptide receptor studies. 14. Stereochemistry determines agonist efficacy and intrinsic efficacy in the [(35)S]GTP-gamma-S functional binding assay.

Probes for narcotic receptor mediated phenomena. 40. N-substituted cis-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-8-ols

Identification of a novel "almost neutral" micro-opioid receptor antagonist in CHO cells expressing the cloned human mu-opioid receptor.

Probes for narcotic receptor mediated phenomena. 37. Synthesis and opioid binding affinity of the final pair of oxide-bridged phenylmorphans, the ortho- and para-b-isomers and their N-phenethyl analogues, and the synthesis of the N-phenethyl analogu

Synthetic studies of neoclerodane diterpenoids from Salvia splendens and evaluation of Opioid Receptor affinity.

Inverse agonists and neutral antagonists at mu opioid receptor (MOR): possible role of basal receptor signaling in narcotic dependence.

Probes for narcotic receptor mediated phenomena. Part 28: new opioid antagonists from enantiomeric analogues of 5-(3-hydroxyphenyl)-N-phenylethylmorphan.

Opioid ligands with mixed properties from substituted enantiomeric N-phenethyl-5-phenylmorphans. Synthesis of a micro-agonist delta-antagonist and delta-inverse agonists.

Investigation of the N-substituent conformation governing potency and mu receptor subtype-selectivity in (+)-(3R, 4R)-dimethyl-4-(3-hydroxyphenyl)piperidine opioid antagonists.

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957-969

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scholarly article

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10.1021/JM1011676

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English

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P478

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Ross W Bittman

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2011-01-19T00:00:00Z

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49767048

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21247164

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3047451

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