Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes.
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Expansion of the alpha 2-adrenergic receptor family: cloning and characterization of a human alpha 2-adrenergic receptor subtype, the gene for which is located on chromosome 2125I-4-(2-[7-amino-2-[2-furyl][1,2,4]triazolo[2,3-a][1,3,5] triazin-5-yl-amino]ethyl)phenol, a high affinity antagonist radioligand selective for the A2a adenosine receptorCloning and expression of a human kidney cDNA for an alpha 2-adrenergic receptor subtypePharmacological actions of the selective and non-selective beta-adrenoceptor antagonists celiprolol, bisoprolol and propranolol on human bronchiNebivolol, bucindolol, metoprolol and carvedilol are devoid of intrinsic sympathomimetic activity in human myocardiumElectrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptorsStructural basis of beta-adrenergic receptor subtype specificity studied with chimeric beta 1/beta 2-adrenergic receptorsAntagonism of thyroid hormone action by amiodarone in rat pituitary tumor cellsChronic caffeine ingestion sensitizes the A1 adenosine receptor-adenylate cyclase system in rat cerebral cortexHigh affinity acylating antagonists for the A1 adenosine receptor: identification of binding subunitRole of the second extracellular loop of adenosine receptors in agonist and antagonist binding. Analysis of chimeric A1/A3 adenosine receptorsThe Influence of the 1-(3-Trifluoromethyl-Benzyl)-1H-Pyrazole-4-yl Moiety on the Adenosine Receptors Affinity Profile of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine DerivativesModulation of the conformational state of the SV2A protein by an allosteric mechanism as evidenced by ligand binding assays.Hyperactivity of the dopaminergic system in NTS1 and NTS2 null mice.Cloning, expression, and characterization of the unique bovine A1 adenosine receptor. Studies on the ligand binding site by site-directed mutagenesisMolecular cloning and expression of the cDNA for the hamster alpha 1-adrenergic receptor.Identification of an adenosine receptor domain specifically involved in binding of 5'-substituted adenosine agonists.Guanine nucleotides modulate the binding affinity of the oligopeptide chemoattractant receptor on human polymorphonuclear leukocytesSimilarities in the behavior and molecular deficits in the frontal cortex between the neurotensin receptor subtype 1 knockout mice and chronic phencyclidine-treated mice: relevance to schizophreniaIdentification of the A2 adenosine receptor binding subunit by photoaffinity crosslinking.An accurate method for determination of receptor-ligand and enzyme-inhibitor dissociation constants from displacement curves.TRIFUNCTIONAL LIGANDS: A RADIOIODINATED HIGH AFFINITY ACYLATING ANTAGONIST FOR THE A1 ADENOSINE RECEPTOR.Direct relationship between mononuclear leukocyte and lung beta-adrenergic receptors and apparent reciprocal regulation of extravascular, but not intravascular, alpha- and beta-adrenergic receptors by the sympathochromaffin system in humans.Multiple components of the A1 adenosine receptor-adenylate cyclase system are regulated in rat cerebral cortex by chronic caffeine ingestion.Pre-beta-very low density lipoproteins as precursors of beta-very low density lipoproteins. A model for the pathogenesis of familial dysbetalipoproteinemia (type III hyperlipoproteinemia)High receptor binding affinity of lipoproteins in atypical dysbetalipoproteinemia (type III hyperlipoproteinemia)Role of thrombospondin in platelet aggregation.Regions of the alpha 1-adrenergic receptor involved in coupling to phosphatidylinositol hydrolysis and enhanced sensitivity of biological functionADP can induce aggregation of human platelets via both P2Y(1) and P(2T) receptors.Human breast cancer cell line MDA-MB-231 expresses endogenous A2B adenosine receptors mediating a Ca2+ signal.Quantification of beta adrenergic receptor subtypes in beta-arrestin knockout mouse airways.High molecular weight kininogen binds to unstimulated plateletsNovel histamine H3 receptor antagonists: affinities in an H3 receptor binding assay and potencies in two functional H3 receptor models.Reduced high-affinity alpha 1-adrenoceptors in liver of senescent rats: implications of assessment at various temperaturesThe palmitoylated cysteine of the cytoplasmic tail of alpha 2A-adrenergic receptors confers subtype-specific agonist-promoted downregulationA chemoattractant receptor on macrophages exists in two affinity states regulated by guanine nucleotides.Glycoprotein nature of the A2-adenosine receptor binding subunitAffinity chromatography of human platelet alpha 2-adrenergic receptors.Purification and characterization of bovine cerebral cortex A1 adenosine receptor.A new high affinity, iodinated adenosine receptor antagonist as a radioligand/photoaffinity crosslinking probe.
P2860
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P2860
Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes.
description
1982 nî lūn-bûn
@nan
1982 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
1982 թվականի հունվարին հրատարակված գիտական հոդված
@hy
1982年の論文
@ja
1982年論文
@yue
1982年論文
@zh-hant
1982年論文
@zh-hk
1982年論文
@zh-mo
1982年論文
@zh-tw
1982年论文
@wuu
name
Validation and statistical ana ...... macological receptor subtypes.
@ast
Validation and statistical ana ...... macological receptor subtypes.
@en
Validation and statistical ana ...... macological receptor subtypes.
@nl
type
label
Validation and statistical ana ...... macological receptor subtypes.
@ast
Validation and statistical ana ...... macological receptor subtypes.
@en
Validation and statistical ana ...... macological receptor subtypes.
@nl
prefLabel
Validation and statistical ana ...... macological receptor subtypes.
@ast
Validation and statistical ana ...... macological receptor subtypes.
@en
Validation and statistical ana ...... macological receptor subtypes.
@nl
P2093
P1476
Validation and statistical ana ...... macological receptor subtypes.
@en
P2093
Hancock AA
Lefkowitz RJ
P577
1982-01-01T00:00:00Z