Exploration of dimensions of estrogen potency: parsing ligand binding and coactivator binding affinities.
about
3D models of MBP, a biologically active metabolite of bisphenol A, in human estrogen receptor α and estrogen receptor βDesign of pathway preferential estrogens that provide beneficial metabolic and vascular effects without stimulating reproductive tissuesComparison of life-stage-dependent internal dosimetry for bisphenol A, ethinyl estradiol, a reference estrogen, and endogenous estradiol to test an estrogenic mode of action in Sprague Dawley rats.Diarylpropionitrile (DPN) enantiomers: synthesis and evaluation of estrogen receptor β-selective ligands.Endocrine-disrupting chemicals and public health protection: a statement of principles from The Endocrine SocietyThe uterine and vascular actions of estetrol delineate a distinctive profile of estrogen receptor α modulation, uncoupling nuclear and membrane activation.Microbiome and malignancyPharmacokinetics of the estrogen receptor subtype-selective ligands, PPT and DPN: quantification using UPLC-ES/MS/MSSelective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast CancerEstrogen receptor alpha somatic mutations Y537S and D538G confer breast cancer endocrine resistance by stabilizing the activating function-2 binding conformation.Thiophene-core estrogen receptor ligands having superagonist activity.Estrogen receptor β (ERβ1) transactivation is differentially modulated by the transcriptional coregulator Tip60 in a cis-acting element-dependent mannerMechanisms enforcing the estrogen receptor β selectivity of botanical estrogens.Early histone modifications in the ventromedial hypothalamus and preoptic area following oestradiol administration.Experimental and computational insights on the recognition mechanism between the estrogen receptor α with bisphenol compounds.Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.Activating ESR1 Mutations Differentially Affect the Efficacy of ER Antagonists.Estrogen receptor alpha/co-activator interaction assay: TR-FRETStructurally Novel Antiestrogens Elicit Differential Responses from Constitutively Active Mutant Estrogen Receptors in Breast Cancer Cells and Tumors.Perfluoro-tert-butyl Homoserine Is a Helix-Promoting, Highly Fluorinated, NMR-Sensitive Aliphatic Amino Acid: Detection of the Estrogen Receptor·Coactivator Protein-Protein Interaction by 19F NMR.Human-relevant potency threshold (HRPT) for ERα agonism.
P2860
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P2860
Exploration of dimensions of estrogen potency: parsing ligand binding and coactivator binding affinities.
description
2011 nî lūn-bûn
@nan
2011 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Exploration of dimensions of e ...... oactivator binding affinities.
@ast
Exploration of dimensions of e ...... oactivator binding affinities.
@en
Exploration of dimensions of e ...... oactivator binding affinities.
@nl
type
label
Exploration of dimensions of e ...... oactivator binding affinities.
@ast
Exploration of dimensions of e ...... oactivator binding affinities.
@en
Exploration of dimensions of e ...... oactivator binding affinities.
@nl
prefLabel
Exploration of dimensions of e ...... oactivator binding affinities.
@ast
Exploration of dimensions of e ...... oactivator binding affinities.
@en
Exploration of dimensions of e ...... oactivator binding affinities.
@nl
P2093
P2860
P356
P1476
Exploration of dimensions of e ...... oactivator binding affinities.
@en
P2093
Jillian R Gunther
John A Katzenellenbogen
Kathryn E Carlson
M Jeyakumar
P2860
P304
12971-12982
P356
10.1074/JBC.M110.205112
P407
P577
2011-02-14T00:00:00Z