Tetrahydropyridine-4-carboxamides as novel, potent transient receptor potential vanilloid 1 (TRPV1) antagonists.
about
Increased function of pronociceptive TRPV1 at the level of the joint in a rat model of osteoarthritis pain.Sulfinate derivatives: dual and versatile partners in organic synthesis.In silico research to assist the investigation of carboxamide derivatives as potent TRPV1 antagonists.Diastereoselective additive trifluoromethylation/halogenation of isoxazole triflones: synthesis of all-carbon-functionalized trifluoromethyl isoxazoline triflonesContributions of central and peripheral TRPV1 receptors to mechanically evoked and spontaneous firing of spinal neurons in inflamed rats.TRPV1 antagonist, A-889425, inhibits mechanotransmission in a subclass of rat primary afferent neurons following peripheral inflammation.Chiral fluorinated α-sulfonyl carbanions: enantioselective synthesis and electrophilic capture, racemization dynamics, and structure.Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors.Synthesis of Aryl Triflones through the Trifluoromethanesulfonylation of Benzynes.Heterocycle-linked phenylbenzyl amides as novel TRPV1 antagonists and their TRPV1 binding modes: constraint-induced enhancement of in vitro and in vivo activities.
P2860
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P2860
Tetrahydropyridine-4-carboxamides as novel, potent transient receptor potential vanilloid 1 (TRPV1) antagonists.
description
2008 nî lūn-bûn
@nan
2008 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@ast
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@en
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@nl
type
label
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@ast
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@en
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@nl
prefLabel
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@ast
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@en
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@nl
P2093
P1476
Tetrahydropyridine-4-carboxami ...... nilloid 1 (TRPV1) antagonists.
@en
P2093
Brian S Brown
Bruce R Bianchi
Carol S Surowy
Chih-Hung Lee
Connie R Faltynek
Guo Zhu Zheng
Heath A McDonald
James S Polakowski
John R Koenig
Kennan C Marsh
P304
P356
10.1016/J.BMC.2008.08.005
P407
P577
2008-08-07T00:00:00Z