Analogues and derivatives of oncrasin-1, a novel inhibitor of the C-terminal domain of RNA polymerase II and their antitumor activities.
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Predictive biomarkers in precision medicine and drug development against lung cancerAntitumor activity of a novel oncrasin analogue is mediated by JNK activation and STAT3 inhibitionProdrug oncrasin-266 improves the stability, pharmacokinetics, and safety of NSC-743380Development of synthetic lethality anticancer therapeutics.Expression of sulfotransferase SULT1A1 in cancer cells predicts susceptibility to the novel anticancer agent NSC-743380Antitumor activity of a novel STAT3 inhibitor and redox modulator in non-small cell lung cancer cellsRAS signaling and anti-RAS therapy: lessons learned from genetically engineered mouse models, human cancer cells, and patient-related studies.Microwave-assisted synthesis of 3-nitroindoles from N-aryl enamines via intramolecular arene-alkene couplingTargeted regulation of PI3K/Akt/mTOR/NF-κB signaling by indole compounds and their derivatives: mechanistic details and biological implications for cancer therapySynthesis, structure-activity relationship studies and biological evaluation of novel 2,5-disubstituted indole derivatives as anticancer agents.Simultaneous determination and validation of oncrasin-266 and its metabolites by HPLC-MS/MS: Application to a pharmacokinetic studySynthesis and antimycobacterial activity of novel thiadiazolylhydrazones of 1-substituted indole-3-carboxaldehydes.Synthesis and biological evaluation of novel 6-hydrazinyl-2,4-bismorpholino pyrimidine and 1,3,5-triazine derivatives as potential antitumor agents.Anti-leukemia activity of NSC-743380 in SULT1A1-expressing acute myeloid leukemia cells is associated with inhibitions of cFLIP expression and PI3K/AKT/mTOR activities.Structure-based design of new poly (ADP-ribose) polymerase (PARP-1) inhibitors.Copper-mediated C3-cyanation of indoles by the combination of amine and ammonium.3-Substituted 2-phenyl-indoles: privileged structures for medicinal chemistry
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P2860
Analogues and derivatives of oncrasin-1, a novel inhibitor of the C-terminal domain of RNA polymerase II and their antitumor activities.
description
2011 nî lūn-bûn
@nan
2011 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Analogues and derivatives of o ...... nd their antitumor activities.
@ast
Analogues and derivatives of o ...... nd their antitumor activities.
@en
Analogues and derivatives of o ...... nd their antitumor activities.
@nl
type
label
Analogues and derivatives of o ...... nd their antitumor activities.
@ast
Analogues and derivatives of o ...... nd their antitumor activities.
@en
Analogues and derivatives of o ...... nd their antitumor activities.
@nl
prefLabel
Analogues and derivatives of o ...... nd their antitumor activities.
@ast
Analogues and derivatives of o ...... nd their antitumor activities.
@en
Analogues and derivatives of o ...... nd their antitumor activities.
@nl
P2093
P2860
P356
P1476
Analogues and derivatives of o ...... nd their antitumor activities.
@en
P2093
Bingliang Fang
Jinsong Liu
Shuhong Wu
Xiaoli Wei
Xiaoying Liu
P2860
P304
P356
10.1021/JM101417N
P407
P577
2011-04-06T00:00:00Z