Discovery of a diaminoquinoxaline benzenesulfonamide antagonist of HIV-1 Nef function using a yeast-based phenotypic screen
about
Dynamics of the Tec-family tyrosine kinase SH3 domains.Subtle Dynamic Changes Accompany Hck Activation by HIV-1 Nef and are Reversed by an Antiretroviral Kinase Inhibitor.Interaction with the Src homology (SH3-SH2) region of the Src-family kinase Hck structures the HIV-1 Nef dimer for kinase activation and effector recruitmentSynthesis and evaluation of orally active small molecule HIV-1 Nef antagonists.Association with PAK2 Enables Functional Interactions of Lentiviral Nef Proteins with the Exocyst Complex.Identification of Binding Mode and Prospective Structural Features of Novel Nef Protein Inhibitors as Potential Anti-HIV Drugs.A Highly Conserved Residue in HIV-1 Nef Alpha Helix 2 Modulates Protein Expression.Imidazoline scaffold in medicinal chemistry: a patent review (2012-2015).Pharmacologic HIV-1 Nef blockade promotes CD8 T cell-mediated elimination of latently HIV-1-infected cells in vitro.Remodeling of HIV-1 Nef Structure by Src-Family Kinase Binding.All-Round Manipulation of the Actin Cytoskeleton by HIV.A single β-octyl glucoside molecule induces HIV-1 Nef dimer formation in the absence of partner protein binding.
P2860
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P2860
Discovery of a diaminoquinoxaline benzenesulfonamide antagonist of HIV-1 Nef function using a yeast-based phenotypic screen
description
2013 nî lūn-bûn
@nan
2013 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
Discovery of a diaminoquinoxal ...... yeast-based phenotypic screen
@en
type
label
Discovery of a diaminoquinoxal ...... yeast-based phenotypic screen
@en
prefLabel
Discovery of a diaminoquinoxal ...... yeast-based phenotypic screen
@en
P2093
P2860
P356
P1433
P1476
Discovery of a diaminoquinoxal ...... yeast-based phenotypic screen
@en
P2093
Billy W Day
Gary Thomas
John Jeff Alvarado
Katelyn Atkins
Laurel Thomas
Lori A Emert-Sedlak
Naveena Yanamala
Purushottam Narute
Ronald P Trible
Thomas E Smithgall
P2860
P2888
P356
10.1186/1742-4690-10-135
P577
2013-11-14T00:00:00Z
P5875
P6179
1022093673