[3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors.
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Non-xanthine heterocycles: activity as antagonists of A1- and A2-adenosine receptorsBinary drugs: conjugates of purines and a peptide that bind to both adenosine and substance P receptorsElectrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptorsPotent convulsant actions of the adenosine receptor antagonist, xanthine amine congener (XAC)High affinity acylating antagonists for the A1 adenosine receptor: identification of binding subunitAdenosine Receptors: The Contributions by John W. Daly.Trifunctional agents as a design strategy for tailoring ligand properties: irreversible inhibitors of A1 adenosine receptors.Biophysical mapping of the adenosine A2A receptorXanthines as adenosine receptor antagonists.Programmable nanoscaffolds that control ligand display to a G-protein-coupled receptor in membranes to allow dissection of multivalent effects.Identification of the A2 adenosine receptor binding subunit by photoaffinity crosslinking.Multiple components of the A1 adenosine receptor-adenylate cyclase system are regulated in rat cerebral cortex by chronic caffeine ingestion.XAC, a functionalized congener of 1,3-dialkylxanthine, antagonizes A1 adenosine receptor-mediated inhibition of renin secretion in vitro.Probing the binding site of the A1 adenosine receptor reengineered for orthogonal recognition by tailored nucleosides.A [3H]amine congener of 1,3-dipropyl-8-phenylxanthine. A new radioligand for A2 adenosine receptors of human platelets.T-cell specific defect in expression of the NTPDase CD39 as a biomarker for lupusMolecular probes for extracellular adenosine receptors.Characterization of human striatal A2-adenosine receptors using radioligand binding and photoaffinity labelingXanthine functionalized congeners as potent ligands at A2-adenosine receptors.Species differences in structure-activity relationships of adenosine agonists and xanthine antagonists at brain A1 adenosine receptors.8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.A new high affinity, iodinated adenosine receptor antagonist as a radioligand/photoaffinity crosslinking probe.Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.[(3)H]XAC (xanthine amine congener) is a radioligand for A(2)-adenosine receptors in rabbit striatum.Frog secretions and hunting magic in the upper Amazon: identification of a peptide that interacts with an adenosine receptor.Analysis of agonist-antagonist interactions at A1 adenosine receptors.Further characterization of the renovascular effects of N6-cyclohexyladenosine in the isolated perfused rat kidney.Affinity chromatography of the bovine cerebral cortex A1 adenosine receptorDemonstration of both A1 and A2 adenosine receptors in DDT1 MF-2 smooth muscle cellsInteraction of dihydropyridine calcium channel agonists and antagonists with adenosine receptors.Penetration of adenosine antagonists into mouse brain as determined by ex vivo binding.KW-3902, a selective high affinity antagonist for adenosine A1 receptors.Apparent heterogeneity of cardiac A1 adenosine receptors as revealed by radioligand binding experiments on N-ethylmaleimide-treated membranes.Bronchodilatory activity and pharmacokinetics of new xanthines in guinea-pigs.Agonists and antagonists recognize different but overlapping populations of A1 adenosine receptors: modulation of receptor number by MgCl2, solubilization, and guanine nucleotides.
P2860
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P2860
[3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors.
description
1986 nî lūn-bûn
@nan
1986年の論文
@ja
1986年論文
@yue
1986年論文
@zh-hant
1986年論文
@zh-hk
1986年論文
@zh-mo
1986年論文
@zh-tw
1986年论文
@wuu
1986年论文
@zh
1986年论文
@zh-cn
name
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@ast
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@en
type
label
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@ast
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@en
prefLabel
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@ast
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@en
P2093
P2860
P356
P1476
[3H]xanthine amine congener of ...... igand for adenosine receptors.
@en
P2093
P2860
P304
P356
10.1073/PNAS.83.11.4089
P407
P577
1986-06-01T00:00:00Z